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Find link is a tool written by Edward Betts.searching for TAAR1 19 found (130 total)
alternate case: tAAR1
Substituted cathinone
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do not act as agonists of the human trace amine-associated receptor 1 (TAAR1). This may potentiate their stimulating and addictive effects. The derivativesReuptake (1,897 words) [view diff] exact match in snippet view article find links to article
It has been shown that AMPH acts upon trace amine-associated receptor 1 (TAAR1) to induce efflux and reuptake inhibition in the serotonin, norepinephrineGlutamate transporter (2,828 words) [view diff] exact match in snippet view article find links to article
PMID 24950453. TAAR1 overexpression significantly decreased EAAT-2 levels and glutamate clearance ... METH treatment activated TAAR1 leading to intracellularBupropion (12,534 words) [view diff] exact match in snippet view article find links to article
showed agonist activity of solriamfetol at human, mouse, and rat TAAR1 receptors. hTAAR1 EC50 values (10–16 μM) were within the clinically observed therapeuticMonoamine transporter (2,342 words) [view diff] exact match in snippet view article find links to article
neurotransmitters. Once inside, it binds to TAAR1 or enters synaptic vesicles through VMAT2. When amphetamine binds to TAAR1, it reduces post-synaptic receptorExcitatory amino acid reuptake inhibitor (479 words) [view diff] exact match in snippet view article find links to article
G, Pouzet B, Bettler B, Caron MG, Wettstein JG, Hoener MC (May 2011). "TAAR1 activation modulates monoaminergic neurotransmission, preventing hyperdopaminergic4-HO-MET (598 words) [view diff] exact match in snippet view article find links to article
Binding sites Binding affinity Ki (μM) 5-HT1A 0.228 5-HT2A 0.057 5-HT2C 0.141 D1 >25 D2 4 D3 6.7 α1A 9.7 α2A 2.4 TAAR1 3.1 H1 0.82 SERT 0.2 DAT >26 NET 135-MeO-MiPT (1,080 words) [view diff] exact match in snippet view article find links to article
Binding Sites Binding Affinity Ki (μM) 5-HT1A 0.058 5-HT2A 0.163 5-HT2C 1.3 D1 >25 D2 >25 D3 >25 α1A >12 α2A 5.3 TAAR1 >15 H1 3.9 SERT 3.3 DAT >26 NET >22Steroid hormone receptor (2,796 words) [view diff] exact match in snippet view article find links to article
binds androgens, and Thyroid Hormone and Trace Amine Associated Receptor 1 (TAAR1) binds Thyroid hormone (though not technically steroid hormones, thyroidList of investigational antidepressants (11,184 words) [view diff] exact match in snippet view article find links to article
receptor 1 (TAAR1) agonist Ulotaront (SEP-363856; SEP-856) – serotonin 5-HT1A receptor agonist and trace amine-associated receptor 1 (TAAR1) agonist PRAX-114Zolmitriptan (1,864 words) [view diff] exact match in snippet view article find links to article
EA, Hanratty L, Koblan KS, Foley A, Dedic N, Bristow LJ (August 2024). "TAAR1 and 5-HT1B receptor agonists attenuate autism-like irritability and aggressionDiPT (587 words) [view diff] exact match in snippet view article find links to article
Binding sites Binding affinity (Ki, μM) 5-HT1A 0.538 5-HT2A 1.2 5-HT2C 6.5 D1 >25 D2 >25 D3 >25 α1A >12 α2A 3.6 TAAR1 >15 H1 0.92 SERT 0.18 DAT 4.1 NET 8.9Substituted β-hydroxyamphetamine (1,363 words) [view diff] exact match in snippet view article find links to article
4-fluoroephedrine are not agonists of the human trace amine-associated receptor 1 (TAAR1). With regard to medical and other uses, β-hydroxyamphetamines are employed5-MeO-aMT (1,159 words) [view diff] exact match in snippet view article find links to article
Binding Sites Binding Affinity Ki (μM) 5-HT1A 0.046 5-HT2A 0.034 5-HT2C 0.09 D1 >25 D2 >25 D3 >25 α1A >12 α2A 11 TAAR1 1.1 H1 >25 SERT 12 DAT >26 NET >22Mescaline (6,052 words) [view diff] exact match in snippet view article find links to article
4–8.9 α2B >10 α2C 0.75 β1 >10 β2 >10 D1 >14 D2 >10 D3 >17 D4 >10 D5 >10 TAAR1 3.3–11 (mouse/rat) I1 2.7 σ1 >10 σ2 >10 SERTTooltip Serotonin transporterMephedrone (12,257 words) [view diff] exact match in snippet view article find links to article
receptors, α2-adrenergic receptors, and trace amine-associated receptor 1 (TAAR1). Mephedrone administration leads to increased extracellular dopamine inPsychedelic drug (9,054 words) [view diff] exact match in snippet view article find links to article
monoamine neurotransmission by binding to trace amine-associated receptor 1 (TAAR1), which plays a significant role in regulating neurotransmission in dopamineSynthetic drug (2,877 words) [view diff] exact match in snippet view article find links to article
negative inotropism in isolated cardiac tissues of rats due to stimulation of TAAR1, which is in contrast with human pharmacology. Alprazolam binds to GABABernard Lerer (1,613 words) [view diff] exact match in snippet view article find links to article
Bernard; Lifschytz, Tzuri (2022). "Role of 5-HT2A, 5-HT2C, 5-HT1A and TAAR1 Receptors in the Head Twitch Response Induced by 5-Hydroxytryptophan and