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searching for TAAR1 19 found (130 total)

alternate case: tAAR1

Substituted cathinone (2,370 words) [view diff] exact match in snippet view article find links to article

do not act as agonists of the human trace amine-associated receptor 1 (TAAR1). This may potentiate their stimulating and addictive effects. The derivatives
Reuptake (1,897 words) [view diff] exact match in snippet view article find links to article
It has been shown that AMPH acts upon trace amine-associated receptor 1 (TAAR1) to induce efflux and reuptake inhibition in the serotonin, norepinephrine
Glutamate transporter (2,828 words) [view diff] exact match in snippet view article find links to article
PMID 24950453. TAAR1 overexpression significantly decreased EAAT-2 levels and glutamate clearance ... METH treatment activated TAAR1 leading to intracellular
Bupropion (12,534 words) [view diff] exact match in snippet view article find links to article
showed agonist activity of solriamfetol at human, mouse, and rat TAAR1 receptors. hTAAR1 EC50 values (10–16 μM) were within the clinically observed therapeutic
Monoamine transporter (2,342 words) [view diff] exact match in snippet view article find links to article
neurotransmitters. Once inside, it binds to TAAR1 or enters synaptic vesicles through VMAT2. When amphetamine binds to TAAR1, it reduces post-synaptic receptor
Excitatory amino acid reuptake inhibitor (479 words) [view diff] exact match in snippet view article find links to article
G, Pouzet B, Bettler B, Caron MG, Wettstein JG, Hoener MC (May 2011). "TAAR1 activation modulates monoaminergic neurotransmission, preventing hyperdopaminergic
4-HO-MET (598 words) [view diff] exact match in snippet view article find links to article
Binding sites Binding affinity Ki (μM) 5-HT1A 0.228 5-HT2A 0.057 5-HT2C 0.141 D1 >25 D2 4 D3 6.7 α1A 9.7 α2A 2.4 TAAR1 3.1 H1 0.82 SERT 0.2 DAT >26 NET 13
5-MeO-MiPT (1,080 words) [view diff] exact match in snippet view article find links to article
Binding Sites Binding Affinity Ki (μM) 5-HT1A 0.058 5-HT2A 0.163 5-HT2C 1.3 D1 >25 D2 >25 D3 >25 α1A >12 α2A 5.3 TAAR1 >15 H1 3.9 SERT 3.3 DAT >26 NET >22
Steroid hormone receptor (2,796 words) [view diff] exact match in snippet view article find links to article
binds androgens, and Thyroid Hormone and Trace Amine Associated Receptor 1 (TAAR1) binds Thyroid hormone (though not technically steroid hormones, thyroid
List of investigational antidepressants (11,184 words) [view diff] exact match in snippet view article find links to article
receptor 1 (TAAR1) agonist Ulotaront (SEP-363856; SEP-856) – serotonin 5-HT1A receptor agonist and trace amine-associated receptor 1 (TAAR1) agonist PRAX-114
Zolmitriptan (1,864 words) [view diff] exact match in snippet view article find links to article
EA, Hanratty L, Koblan KS, Foley A, Dedic N, Bristow LJ (August 2024). "TAAR1 and 5-HT1B receptor agonists attenuate autism-like irritability and aggression
DiPT (587 words) [view diff] exact match in snippet view article find links to article
Binding sites Binding affinity (Ki, μM) 5-HT1A 0.538 5-HT2A 1.2 5-HT2C 6.5 D1 >25 D2 >25 D3 >25 α1A >12 α2A 3.6 TAAR1 >15 H1 0.92 SERT 0.18 DAT 4.1 NET 8.9
Substituted β-hydroxyamphetamine (1,363 words) [view diff] exact match in snippet view article find links to article
4-fluoroephedrine are not agonists of the human trace amine-associated receptor 1 (TAAR1). With regard to medical and other uses, β-hydroxyamphetamines are employed
5-MeO-aMT (1,159 words) [view diff] exact match in snippet view article find links to article
Binding Sites Binding Affinity Ki (μM) 5-HT1A 0.046 5-HT2A 0.034 5-HT2C 0.09 D1 >25 D2 >25 D3 >25 α1A >12 α2A 11 TAAR1 1.1 H1 >25 SERT 12 DAT >26 NET >22
Mescaline (6,052 words) [view diff] exact match in snippet view article find links to article
4–8.9 α2B >10 α2C 0.75 β1 >10 β2 >10 D1 >14 D2 >10 D3 >17 D4 >10 D5 >10 TAAR1 3.3–11 (mouse/rat) I1 2.7 σ1 >10 σ2 >10 SERTTooltip Serotonin transporter
Mephedrone (12,257 words) [view diff] exact match in snippet view article find links to article
receptors, α2-adrenergic receptors, and trace amine-associated receptor 1 (TAAR1). Mephedrone administration leads to increased extracellular dopamine in
Psychedelic drug (9,054 words) [view diff] exact match in snippet view article find links to article
monoamine neurotransmission by binding to trace amine-associated receptor 1 (TAAR1), which plays a significant role in regulating neurotransmission in dopamine
Synthetic drug (2,877 words) [view diff] exact match in snippet view article find links to article
negative inotropism in isolated cardiac tissues of rats due to stimulation of TAAR1, which is in contrast with human pharmacology. Alprazolam binds to GABA
Bernard Lerer (1,613 words) [view diff] exact match in snippet view article find links to article
Bernard; Lifschytz, Tzuri (2022). "Role of 5-HT2A, 5-HT2C, 5-HT1A and TAAR1 Receptors in the Head Twitch Response Induced by 5-Hydroxytryptophan and