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Longer titles found: Bioorganic & Medicinal Chemistry Letters (view)

searching for Bioorganic & Medicinal Chemistry 522 found (936 total)

alternate case: bioorganic & Medicinal Chemistry

8-Carboxamidocyclazocine (623 words) [view diff] exact match in snippet view article find links to article

structure-activity relationships of 2,6-methano-3-benzazocines". Bioorganic & Medicinal Chemistry Letters. 11 (5): 623–6. doi:10.1016/S0960-894X(01)00014-2.

LeDock (757 words) [view diff] exact match in snippet view article find links to article

conformation of its kinase domain generated by molecular dynamics". Bioorganic & Medicinal Chemistry Letters. 23 (20): 5721–5726. doi:10.1016/j.bmcl.2013.08.009

QMPSB (497 words) [view diff] exact match in snippet view article find links to article

ligands: identification of a lead and initial SAR studies". Bioorganic & Medicinal Chemistry Letters. 17 (1): 272–7. doi:10.1016/j.bmcl.2006.09.049. PMID 17027269

List of JWH cannabinoids (883 words) [view diff] exact match in snippet view article find links to article

substituents. New highly selective CB(2) receptor agonists". Bioorganic & Medicinal Chemistry. 13 (1): 89–112. doi:10.1016/j.bmc.2004.09.050. PMID 15582455

Metabotropic glutamate receptor 2 (2,647 words) [view diff] exact match in snippet view article find links to article

selective, orally bioavailable positive modulators of mGluR2". Bioorganic & Medicinal Chemistry Letters. 20 (2): 759–62. doi:10.1016/j.bmcl.2009.11.032. PMID 20005096

Unifiram (648 words) [view diff] exact match in snippet view article find links to article

(DM235), two novel and potent cognition enhancing drugs". Bioorganic & Medicinal Chemistry. 12 (1): 71–85. doi:10.1016/j.bmc.2003.10.025. PMID 14697772

KM-233 (476 words) [view diff] exact match in snippet view article find links to article

substituted side-chain analogues of classical cannabinoids". Bioorganic & Medicinal Chemistry Letters. 13 (20): 3487–90. doi:10.1016/s0960-894x(03)00729-7

Salvinorin (735 words) [view diff] exact match in snippet view article find links to article

and selective κ opioids: salvinorin B alkoxymethyl ethers". Bioorganic & Medicinal Chemistry. 16 (3): 1279–86. doi:10.1016/j.bmc.2007.10.067. PMC 2568987

5-HT6 receptor (3,308 words) [view diff] exact match in snippet view article find links to article

as selective brain penetrant 5-HT6 receptor antagonists". Bioorganic & Medicinal Chemistry Letters. 18 (20): 5698–700. doi:10.1016/j.bmcl.2008.08.010

Efaroxan (300 words) [view diff] exact match in snippet view article find links to article

Imbert, T. (1999). "A new efficient synthesis of efaroxan". Bioorganic & Medicinal Chemistry Letters 9 (20): 3021–3022. doi:10.1016/S0960-894X(99)00531-4

Fiesselmann thiophene synthesis (843 words) [view diff] exact match in snippet view article find links to article

arthritis and osteoporosis: thienyl, furyl, and pyrrolyl ureas". Bioorganic & Medicinal Chemistry Letters. 11 (1): 9–12. doi:10.1016/S0960-894X(00)00574-6. PMID 11140741

Hypocretin (orexin) receptor 2 (1,672 words) [view diff] exact match in snippet view article

potent and selective orexin receptor 2 (OX(2)R) antagonists". Bioorganic & Medicinal Chemistry Letters. 14 (16): 4225–4229. doi:10.1016/j.bmcl.2004.06.032

Dihydrostilbenoid (572 words) [view diff] exact match in snippet view article find links to article

(2010). "Dihydro-resveratrol—A potent dietary polyphenol". Bioorganic & Medicinal Chemistry Letters. 20 (20): 6149–51. doi:10.1016/j.bmcl.2010.08.002.

LBP-1 (drug) (284 words) [view diff] exact match in snippet view article

of indole-3-heterocycles as agonists of the CB1 receptor". Bioorganic & Medicinal Chemistry Letters. 21 (1): 506–9. doi:10.1016/j.bmcl.2010.10.093. PMID 21075630

MN-25 (854 words) [view diff] exact match in snippet view article find links to article

2002). "C-3 Amido-indole cannabinoid receptor modulators". Bioorganic & Medicinal Chemistry Letters. 12 (17): 2399–402. doi:10.1016/S0960-894X(02)00466-3

L-371,257 (442 words) [view diff] exact match in snippet view article find links to article

L-371,257 containing a 1-R-(pyridyl)ethyl ether terminus". Bioorganic & Medicinal Chemistry Letters. 8 (21): 3081–6. doi:10.1016/S0960-894X(98)00568-X

VU-0238429 (263 words) [view diff] exact match in snippet view article find links to article

heterobiaryl ether derived M5 positive allosteric modulators". Bioorganic & Medicinal Chemistry Letters. 20 (19): 5617–5622. doi:10.1016/j.bmcl.2010.08.042

(+)-CPCA (4,041 words) [view diff] exact match in snippet view article

binding properties of (R)-2β,3β- and (R)-2α,3α-diaryltropanes". Bioorganic & Medicinal Chemistry Letters. 8 (24): 3689–92. doi:10.1016/s0960-894x(98)00673-8

Epiboxidine (477 words) [view diff] exact match in snippet view article find links to article

neuronal nicotinic acetylcholine receptor subtypes" (PDF). Bioorganic & Medicinal Chemistry Letters. 18 (16): 4651–4. doi:10.1016/j.bmcl.2008.07.016. hdl:2434/59291

Himbacine (243 words) [view diff] exact match in snippet view article find links to article

Discovery of a Pharmacophoric Element for M2-Selectivity". Bioorganic & Medicinal Chemistry Letters. 5 (1): 61–66. doi:10.1016/0960-894X(94)00459-S. Chackalamannil

9-Aminomethyl-9,10-dihydroanthracene (385 words) [view diff] exact match in snippet view article find links to article

spiro[9,10-dihydroanthracene]-9,3(')-pyrrolidine (SpAMDA)". Bioorganic & Medicinal Chemistry Letters. 14 (9): 2279–83. doi:10.1016/j.bmcl.2004.02.014. PMID 15081025

CX717 (1,512 words) [view diff] exact match in snippet view article find links to article

potent positive allosteric AMPA receptor modulators: part I". Bioorganic & Medicinal Chemistry Letters. 21 (13): 3923–3926. doi:10.1016/j.bmcl.2011.05.026

Fenobam (839 words) [view diff] exact match in snippet view article find links to article

structure-activity relationship study of fenobam analogues". Bioorganic & Medicinal Chemistry Letters. 16 (5): 1142–5. doi:10.1016/j.bmcl.2005.11.092. PMID 16380255

Biphalin (524 words) [view diff] exact match in snippet view article find links to article

analogues of the potent dimeric opioid peptide, biphalin". Bioorganic & Medicinal Chemistry Letters. 9 (18): 2763–6. doi:10.1016/S0960-894X(99)00464-3

Adenosine A2B receptor (2,125 words) [view diff] exact match in snippet view article find links to article

affinity and selective A2B adenosine receptor antagonists". Bioorganic & Medicinal Chemistry Letters. 16 (2): 302–306. doi:10.1016/j.bmcl.2005.10.002. PMID 16275090

Ro67-4853 (335 words) [view diff] exact match in snippet view article find links to article

as potent, orally available mGlu1 receptor enhancers". Bioorganic & Medicinal Chemistry Letters. 15 (20): 4628–31. doi:10.1016/j.bmcl.2005.05.135.

Conessine (336 words) [view diff] exact match in snippet view article find links to article

steroidal alkaloids from Funtumia elastica (Preuss) Stapf". Bioorganic & Medicinal Chemistry Letters. 15 (10): 2637–40. doi:10.1016/j.bmcl.2005.03.021.

Phellinus (482 words) [view diff] exact match in snippet view article find links to article

antioxidants in the medicinal mushrooms Inonotus and Phellinus". Bioorganic & Medicinal Chemistry. 15 (10): 3309–14. doi:10.1016/j.bmc.2007.03.039. PMID 17387019

Isonotholaenic acid (136 words) [view diff] exact match in snippet view article find links to article

System. A New Skeletal Basis for Antiplasmodial Compounds". Bioorganic & Medicinal Chemistry Letters. 13 (16): 2769–2772. doi:10.1016/S0960-894X(03)00509-2

Metabotropic glutamate receptor 3 (3,074 words) [view diff] exact match in snippet view article find links to article

acid and its 6-heptyl ester, a potent mGluR2 antagonist". Bioorganic & Medicinal Chemistry. 16 (8): 4359–66. doi:10.1016/j.bmc.2008.02.066. PMID 18348906

4-Fluoromethylphenidate (513 words) [view diff] exact match in snippet view article find links to article

binding affinities at dopamine and serotonin transport sites". Bioorganic & Medicinal Chemistry Letters. 14 (7): 1799–802. doi:10.1016/j.bmcl.2003.12.097.

Discovery and development of TRPV1 antagonists (4,635 words) [view diff] exact match in snippet view article find links to article

onylamino)benzyl]thiourea analogues as TRPV1 antagonists". Bioorganic & Medicinal Chemistry Letters. 15 (18): 4136–42. doi:10.1016/j.bmcl.2005.06.009.

Cook–Heilbron thiazole synthesis (904 words) [view diff] exact match in snippet view article find links to article

thiazolyl bisamide CSF-1R inhibitors for the treatment of cancer". Bioorganic & Medicinal Chemistry Letters. 18 (17): 4794–4797. doi:10.1016/j.bmcl.2008.07.093

Canadine (633 words) [view diff] exact match in snippet view article find links to article

activities of canadine: Biological effects and structural aspects". Bioorganic & Medicinal Chemistry. 16 (7): 3641–51. doi:10.1016/j.bmc.2008.02.015. PMID 18295494

Lipophilic efficiency (649 words) [view diff] exact match in snippet view article find links to article

synthesis protocols: A Lipophilic Efficiency (LipE) analysis". Bioorganic & Medicinal Chemistry Letters. 19 (15): 4406–9. doi:10.1016/j.bmcl.2009.05.062. PMID 19500981

Butyltolylquinuclidine (136 words) [view diff] exact match in snippet view article find links to article

quinuclidines as a novel class of dopamine transporter inhibitors". Bioorganic & Medicinal Chemistry. 11 (6): 1123–36. doi:10.1016/S0968-0896(02)00450-9. PMID 12614900

Salvinorin A (3,732 words) [view diff] exact match in snippet view article find links to article

their binding affinities for human kappa opioid receptors". Bioorganic & Medicinal Chemistry. 13 (19): 5635–5639. doi:10.1016/j.bmc.2005.05.054. PMID 16084728

CECXG (258 words) [view diff] exact match in snippet view article find links to article

selective antagonists of metabotropic glutamate receptors". Bioorganic & Medicinal Chemistry Letters. 8 (20): 2849–2854. doi:10.1016/S0960-894X(98)00510-1

Benzodioxan (345 words) [view diff] exact match in snippet view article find links to article

potential immunosuppressive agents against RAW264.7 cells". Bioorganic & Medicinal Chemistry. 19 (16): 4895–4902. doi:10.1016/j.bmc.2011.06.061. ISSN 1464-3391

Aglaia (1,032 words) [view diff] exact match in snippet view article find links to article

advances in the biology and chemistry of the flavaglines". Bioorganic & Medicinal Chemistry. 20 (6): 1857–1864. doi:10.1016/j.bmc.2011.10.048. ISSN 0968-0896

Portmanteau inhibitor (199 words) [view diff] exact match in snippet view article find links to article

caffeoyl-anilides as portmanteau inhibitors of HIV-1 integrase and CCR5". Bioorganic & Medicinal Chemistry. 19 (3): 1256–63. doi:10.1016/j.bmc.2010.12.031. PMID 21227704

Alpha-7 nicotinic receptor (2,722 words) [view diff] exact match in snippet view article find links to article

quinuclidines as selective alpha 7 nicotinic receptor ligands". Bioorganic & Medicinal Chemistry Letters. 15 (8): 2073–7. doi:10.1016/j.bmcl.2005.02.045. PMID 15808471

Katherine Seley-Radtke (2,015 words) [view diff] exact match in snippet view article find links to article

analogues and evaluation in the nucleocapsid protein of HIV-1". Bioorganic & Medicinal Chemistry. 27 (13): 2883–92. doi:10.1016/j.bmc.2019.05.019. PMC 6556414

Serotonin–norepinephrine reuptake inhibitor (8,171 words) [view diff] exact match in snippet view article find links to article

multi-target inhibitors as potential agents for depression". Bioorganic & Medicinal Chemistry. 17 (19): 6890–6897. doi:10.1016/j.bmc.2009.08.025. PMID 19740668

Selective progesterone receptor modulator (5,150 words) [view diff] exact match in snippet view article find links to article

as potent and selective progesterone receptor antagonists". Bioorganic & Medicinal Chemistry Letters. 17 (9): 2531–4. doi:10.1016/j.bmcl.2007.02.013. PMID 17317167

Fospropofol (396 words) [view diff] exact match in snippet view article find links to article

propofol analogues with intravenous anaesthetic activity". Bioorganic & Medicinal Chemistry Letters. 11 (7): 927–930. doi:10.1016/S0960-894X(01)00088-9

William Summer Johnson (256 words) [view diff] exact match in snippet view article find links to article

"Tetrahedron Prize for Creativity in Organic Chemistry or Bioorganic & Medicinal Chemistry". Elsevier. Archived from the original on 9 September 2014

Capromorelin (631 words) [view diff] exact match in snippet view article find links to article

characterization of capromorelin analogues with extended half-lives". Bioorganic & Medicinal Chemistry Letters. 12 (22): 3279–82. doi:10.1016/s0960-894x(02)00734-5

BIBP-3226 (472 words) [view diff] exact match in snippet view article find links to article

neuropeptide Y Y1 receptor antagonists related to BIBP 3226". Bioorganic & Medicinal Chemistry Letters. 10 (14): 1597–600. doi:10.1016/S0960-894X(00)00292-4

CCR5 receptor antagonist (5,518 words) [view diff] exact match in snippet view article find links to article

substituted 1-(3,3-diphenylpropyl)-piperidinyl phenylacetamides". Bioorganic & Medicinal Chemistry Letters. 15 (22): 5012–5. doi:10.1016/j.bmcl.2005.08.014. PMID 16154744

Chalconoid (316 words) [view diff] exact match in snippet view article find links to article

chalcone as new class voltage-dependent K+ channel blocker". Bioorganic & Medicinal Chemistry Letters. 18 (1): 137–140. doi:10.1016/j.bmcl.2007.10.114. PMID 18032041

Emma Parmee (722 words) [view diff] exact match in snippet view article find links to article

507: A subnanomolar human β 3 adrenergic receptor agonist". Bioorganic & Medicinal Chemistry Letters. 8 (9): 1107–1112. doi:10.1016/s0960-894x(98)00170-x

Baicalein (477 words) [view diff] exact match in snippet view article find links to article

reticulocyte 15-human and platelet 12-human lipoxygenases". Bioorganic & Medicinal Chemistry. 14 (12): 4295–4301. doi:10.1016/j.bmc.2006.01.057. PMID 16500106

Eudistomin (723 words) [view diff] exact match in snippet view article find links to article

synthesis of eudistomin U and evaluation of its cytotoxicity". Bioorganic & Medicinal Chemistry Letters. 24 (15): 3549–3551. doi:10.1016/j.bmcl.2014.05.049

Diazirine (2,590 words) [view diff] exact match in snippet view article find links to article

M. (2012-01-15). "Diazirine based photoaffinity labeling". Bioorganic & Medicinal Chemistry. Chemical Proteomics. 20 (2): 554–570. doi:10.1016/j.bmc.2011

Streptomyces microflavus (519 words) [view diff] exact match in snippet view article find links to article

insecticidal bioactivity from Streptomyces microflavus neau3". Bioorganic & Medicinal Chemistry Letters. 21 (18): 5145–5148. doi:10.1016/j.bmcl.2011.07.070

CBS-0550 (171 words) [view diff] exact match in snippet view article find links to article

CB2 cannabinoid receptor agonists with an analgesic action". Bioorganic & Medicinal Chemistry. 16 (3): 1111–24. doi:10.1016/j.bmc.2007.10.087. PMID 18006322

Streptomyces atratus (377 words) [view diff] exact match in snippet view article find links to article

"Hydrazidomycins, cytotoxic alkylhydrazides from Streptomyces atratus". Bioorganic & Medicinal Chemistry Letters. 21 (19): 5839–5841. doi:10.1016/j.bmcl.2011.07.108

Fumagillin (1,037 words) [view diff] exact match in snippet view article find links to article

activities of novel, orally available fumagillin analogs". Bioorganic & Medicinal Chemistry Letters Vol. 19 Nr. 17 (2009), blz. 5128-5131 Arico-Muendel

Azaprocin (859 words) [view diff] exact match in snippet view article find links to article

Effects on mu-affinity of arylalkenyl chain modifications". Bioorganic & Medicinal Chemistry. 10 (6): 1929–37. doi:10.1016/s0968-0896(01)00436-9. PMID 11937351

Pyrazolone (512 words) [view diff] exact match in snippet view article find links to article

1-phenyl-3-methyl-5-pyrazolone (PMP), also known as edaravone". Bioorganic & Medicinal Chemistry. 28 (10): 115463. doi:10.1016/j.bmc.2020.115463. PMID 32241621

Cereblon E3 ligase modulator (5,487 words) [view diff] exact match in snippet view article find links to article

October 2003). "α-Fluoro-substituted thalidomide analogues". Bioorganic & Medicinal Chemistry Letters. 13 (20): 3415–3417. doi:10.1016/S0960-894X(03)00778-9

DPA-713 (460 words) [view diff] exact match in snippet view article find links to article

potent ligands for the 18 kDa translocator protein (TSPO)". Bioorganic & Medicinal Chemistry Letters. 20 (19): 5799–802. doi:10.1016/j.bmcl.2010.07.135

Falintolol (57 words) [view diff] exact match in snippet view article find links to article

characterization as beta-adrenergic receptor antagonists". Bioorganic & Medicinal Chemistry. 6 (4): 401–8. doi:10.1016/s0968-0896(97)10051-7. PMID 9597184

J-113,397 (874 words) [view diff] exact match in snippet view article find links to article

the first non-peptide ORL-1 receptor antagonist". Bioorganic & Medicinal Chemistry. 9 (7): 1871–7. doi:10.1016/s0968-0896(01)00085-2. PMID 11425589

Discovery and development of dipeptidyl peptidase-4 inhibitors (5,080 words) [view diff] exact match in snippet view article find links to article

derivatives as dipeptidyl peptidase IV (DPP-IV) inhibitors", Bioorganic & Medicinal Chemistry Letters, 17 (9): 2622–2628, doi:10.1016/j.bmcl.2007.01.111

Samidorphan (994 words) [view diff] exact match in snippet view article find links to article

"Syntheses of novel high affinity ligands for opioid receptors". Bioorganic & Medicinal Chemistry Letters. 19 (8): 2289–2294. doi:10.1016/j.bmcl.2009.02.078

MS-245 (299 words) [view diff] exact match in snippet view article find links to article

"N1-(Benzenesulfonyl)tryptamines as novel 5-HT6 antagonists". Bioorganic & Medicinal Chemistry Letters. 10 (20): 2295–9. doi:10.1016/S0960-894X(00)00453-4

Halijah Ibrahim (368 words) [view diff] exact match in snippet view article find links to article

Boesenbergia rotunda (L.), towards dengue-2 virus NS3 protease. Bioorganic & Medicinal Chemistry Letters 16 3337-3340 "Profile: Halijah Ibrahim". ResearchGate

Tropoxane (561 words) [view diff] exact match in snippet view article find links to article

inhibition of binding at the dopamine and serotonin transporters". Bioorganic & Medicinal Chemistry Letters. 9 (6): 857–62. doi:10.1016/s0960-894x(99)00098-0.

Bafetinib (733 words) [view diff] exact match in snippet view article find links to article

3-substituted benzamide derivatives as Bcr-Abl kinase inhibitors". Bioorganic & Medicinal Chemistry Letters. 16 (5): 1421–5. doi:10.1016/j.bmcl.2005.11.042. PMID 16332440

6,6'-Bieckol (116 words) [view diff] exact match in snippet view article find links to article

phloroglucinol derivative, 6,6′-bieckol, from Ecklonia cava". Bioorganic & Medicinal Chemistry. 16 (17): 7921–7926. doi:10.1016/j.bmc.2008.07.078. PMID 18693022

SYM-2081 (338 words) [view diff] exact match in snippet view article find links to article

selective ligand at the kainate subtype of glutamate receptors". Bioorganic & Medicinal Chemistry Letters. 5 (17): 1973–1976. doi:10.1016/0960-894x(95)00335-q

Org 28312 (278 words) [view diff] exact match in snippet view article find links to article

indole-3-carboxamides as novel CB1 cannabinoid receptor agonists". Bioorganic & Medicinal Chemistry Letters. 20 (16): 4918–21. doi:10.1016/j.bmcl.2010.06.067.

Bcr-Abl tyrosine-kinase inhibitor (6,470 words) [view diff] exact match in snippet view article find links to article

3-substituted benzamide derivatives as Bcr-Abl kinase inhibitors". Bioorganic & Medicinal Chemistry Letters. 16 (5): 1421–1425. doi:10.1016/j.bmcl.2005.11.042

Renin inhibitor (4,784 words) [view diff] exact match in snippet view article find links to article

optimization of renin inhibitors: Orally bioavailable alkyl amines". Bioorganic & Medicinal Chemistry Letters. 19 (13): 3541–3545. doi:10.1016/j.bmcl.2009.04.140

Cutamesine (1,430 words) [view diff] exact match in snippet view article find links to article

selectivity for sigma receptors and monoamine transporters". Bioorganic & Medicinal Chemistry. 23 (1): 222–230. doi:10.1016/j.bmc.2014.11.007. PMC 4274187

AZ-11713908 (315 words) [view diff] exact match in snippet view article find links to article

2008). "5-Sulfonyl-benzimidazoles as selective CB2 agonists". Bioorganic & Medicinal Chemistry Letters. 18 (8): 2574–9. doi:10.1016/j.bmcl.2008.03.048. PMID 18394887

DOB-FLY (345 words) [view diff] exact match in snippet view article find links to article

5-HT2A receptor agonists with ocular hypotensive activity". Bioorganic & Medicinal Chemistry Letters. 17 (11): 2998–3002. doi:10.1016/j.bmcl.2007.03.073

TMC-647055 (196 words) [view diff] exact match in snippet view article find links to article

indole-based macrocycle leading to the discovery of TMC647055". Bioorganic & Medicinal Chemistry Letters. 22 (13): 4437–43. doi:10.1016/j.bmcl.2012.04.113.

Herkinorin (662 words) [view diff] exact match in snippet view article find links to article

diterpenes from Salvia divinorum: exploration of the 1-position". Bioorganic & Medicinal Chemistry Letters. 17 (22): 6111–5. doi:10.1016/j.bmcl.2007.09.050. PMC 2111044

Higenamine (1,611 words) [view diff] exact match in snippet view article find links to article

and structure-activity correlations with related alkaloids". Bioorganic & Medicinal Chemistry. 13 (2): 443–8. doi:10.1016/j.bmc.2004.10.020. PMID 15598565

Remimazolam (1,166 words) [view diff] exact match in snippet view article find links to article

novel ultrashort-acting benzodiazepine receptor agonists". Bioorganic & Medicinal Chemistry Letters. 12 (21): 3215–3218. doi:10.1016/s0960-894x(02)00512-7

Dimiracetam (195 words) [view diff] exact match in snippet view article find links to article

derivatives useful for the treatment of neuropathic pain". Bioorganic & Medicinal Chemistry. 16 (6): 3224–32. doi:10.1016/j.bmc.2007.12.015. PMID 18171618

Rev (HIV) (3,100 words) [view diff] exact match in snippet view article

mismatch-binding ligands as inhibitors for Rev-RRE interaction". Bioorganic & Medicinal Chemistry. 14 (15): 5384–8. doi:10.1016/j.bmc.2006.03.038. PMID 16603366

Ethephon (398 words) [view diff] exact match in snippet view article find links to article

Inhibitors: 2-Chloro-1-(substituted-phenyl)ethylphosphonic Acids". Bioorganic & Medicinal Chemistry. 10 (5): 1281–1290. doi:10.1016/s0968-0896(01)00391-1. PMID 11886791

Melatonin receptor 1B (1,644 words) [view diff] exact match in snippet view article find links to article

derivatives as new selective MT2 melatoninergic ligands". Bioorganic & Medicinal Chemistry. 11 (5): 753–59. doi:10.1016/S0968-0896(02)00473-X. PMID 12538005

Curculigoside (185 words) [view diff] exact match in snippet view article find links to article

(2008). "New polyphenols active on β-amyloid aggregation". Bioorganic & Medicinal Chemistry Letters. 18 (2): 828–31. doi:10.1016/j.bmcl.2007.11.028. PMID 18042380

Discovery and development of non-nucleoside reverse-transcriptase inhibitors (4,737 words) [view diff] exact match in snippet view article find links to article

"The search for potent, small molecule NNRTIs: A review". Bioorganic & Medicinal Chemistry. 17 (16): 5744–62. doi:10.1016/j.bmc.2009.06.060. PMID 19632850

Osanetant (980 words) [view diff] exact match in snippet view article find links to article

1996). "A reliable and efficient synthesis of SR 142801". Bioorganic & Medicinal Chemistry Letters. 6 (19): 2307–2310. doi:10.1016/0960-894X(96)00419-2

Fatty-acid amide hydrolase 1 (3,460 words) [view diff] exact match in snippet view article find links to article

inhibitors. Surprising selectivity of chiral azetidine ureas". Bioorganic & Medicinal Chemistry Letters. 19 (15): 4241–4244. doi:10.1016/j.bmcl.2009.05.097

Curculigoside (185 words) [view diff] exact match in snippet view article find links to article

(2008). "New polyphenols active on β-amyloid aggregation". Bioorganic & Medicinal Chemistry Letters. 18 (2): 828–31. doi:10.1016/j.bmcl.2007.11.028. PMID 18042380

Dieckol (327 words) [view diff] exact match in snippet view article find links to article

phlorotannins from Eisenia bicyclis with BACE1 inhibitory activity". Bioorganic & Medicinal Chemistry Letters. 20 (11): 3211–5. doi:10.1016/j.bmcl.2010.04.093. PMID 20462757

Fuculose (171 words) [view diff] exact match in snippet view article find links to article

"Efficient enzymatic synthesis of L-rhamnulose and L-fuculose". Bioorganic & Medicinal Chemistry Letters. 26 (3): 969–972. doi:10.1016/j.bmcl.2015.12.051. PMC 5984655

CGS-13767 (55 words) [view diff] exact match in snippet view article find links to article

A new class of GABAA brain receptor ligands". Bioorganic & Medicinal Chemistry Letters. 10 (24): 2723–2726. doi:10.1016/S0960-894X(00)00550-3

SQ109 (320 words) [view diff] exact match in snippet view article find links to article

of carbamate prodrugs of SQ109 as antituberculosis agents". Bioorganic & Medicinal Chemistry Letters. 19 (10): 2808–10. doi:10.1016/j.bmcl.2009.03.091.

AM-679 (FLAP inhibitor) (170 words) [view diff] exact match in snippet view article

2-dimethyl-propionic acid (AM679)--a potent FLAP inhibitor". Bioorganic & Medicinal Chemistry Letters. 20 (1): 213–217. doi:10.1016/j.bmcl.2009.10.131. PMID 19914828

HDMP-28 (535 words) [view diff] exact match in snippet view article find links to article

binding affinities at dopamine and serotonin transport sites". Bioorganic & Medicinal Chemistry Letters. 14 (7): 1799–802. doi:10.1016/j.bmcl.2003.12.097.

Fluorenol (687 words) [view diff] exact match in snippet view article find links to article

for next generation modafinil, lessons learned: Part III". Bioorganic & Medicinal Chemistry Letters. 22 (11): 3751–3753. doi:10.1016/j.bmcl.2012.04.031

2C-B-FLY (1,469 words) [view diff] exact match in snippet view article find links to article

the 6-position: effects on 5-HT(2A/2C) receptor affinity". Bioorganic & Medicinal Chemistry Letters. 12 (15): 1997–9. CiteSeerX 10.1.1.688.9483. doi:10

Dinoxyline (156 words) [view diff] exact match in snippet view article find links to article

affinity and potent agonist at all dopamine receptor isoforms". Bioorganic & Medicinal Chemistry. 12 (6): 1403–12. doi:10.1016/j.bmc.2004.01.008. PMID 15018913

O-4210 (195 words) [view diff] exact match in snippet view article find links to article

binding affinity for the dopamine and serotonin transporters". Bioorganic & Medicinal Chemistry. 15 (2): 1067–82. doi:10.1016/j.bmc.2006.10.016. PMC 1829488

Myxopyronin (717 words) [view diff] exact match in snippet view article find links to article

inhibitors of RNA polymerase, synthesis and biological evaluation". Bioorganic & Medicinal Chemistry Letters. 14 (22): 5667–5672. doi:10.1016/j.bmcl.2004.08.045

Oxaprostaglandin (226 words) [view diff] exact match in snippet view article find links to article

as antiglaucoma agents: Synthesis and biological activity". Bioorganic & Medicinal Chemistry. 17 (2): 576–584. doi:10.1016/j.bmc.2008.11.070. PMID 19101156

Mazapertine (477 words) [view diff] exact match in snippet view article find links to article

mazapertine: High affinity ligands for the 5-HT1A receptor". Bioorganic & Medicinal Chemistry Letters. 7 (7): 763. doi:10.1016/S0960-894X(97)00074-7. Reitz

Setrobuvir (169 words) [view diff] exact match in snippet view article find links to article

and orally bioavailable inhibitors of HCV NS5B polymerase". Bioorganic & Medicinal Chemistry Letters. 19 (22): 6404–12. doi:10.1016/j.bmcl.2009.09.045.

Adenosine A2A receptor (5,148 words) [view diff] exact match in snippet view article find links to article

synthesis of thieno[3,2-d]pyrimidine-4-methanone derivatives". Bioorganic & Medicinal Chemistry Letters. 18 (9): 2916–9. doi:10.1016/j.bmcl.2008.03.075. PMID 18406614

Argiotoxin (1,477 words) [view diff] exact match in snippet view article find links to article

AMPA receptors: a perspective on subtype-selective ligands". Bioorganic & Medicinal Chemistry. 18 (4): 1381–1387. doi:10.1016/j.bmc.2009.12.072. ISSN 1464-3391

Enediyne (1,736 words) [view diff] exact match in snippet view article find links to article

microbial genomics to discover new anticancer drug leads". Bioorganic & Medicinal Chemistry Letters. 25 (1): 9–15. doi:10.1016/j.bmcl.2014.11.019. PMC 4480864

Anagliptin (161 words) [view diff] exact match in snippet view article find links to article

hydrochloride salt) as a potent and selective DPP-IV inhibitor". Bioorganic & Medicinal Chemistry. 19 (23): 7221–7. doi:10.1016/j.bmc.2011.09.043. PMID 22019046

Discovery and development of gliflozins (3,188 words) [view diff] exact match in snippet view article find links to article

Jiwen (2011). "Discovery of non-glucoside SGLT2 inhibitors". Bioorganic & Medicinal Chemistry Letters. 21 (8): 2472–2475. doi:10.1016/j.bmcl.2011.02.056

Tebanicline (997 words) [view diff] exact match in snippet view article find links to article

5-Dihydro-1H-pyrrol-2-ylmethoxy)pyridines: synthesis and analgesic activity". Bioorganic & Medicinal Chemistry Letters. 15 (6): 1637–40. doi:10.1016/j.bmcl.2005.01.058. PMID 15745813

Pyrrole–imidazole polyamides (128 words) [view diff] exact match in snippet view article find links to article

binding Pyrrole–imidazole polyamides and their applications". Bioorganic & Medicinal Chemistry. 26 (8): 1393–1411. doi:10.1016/j.bmc.2018.01.026. PMID 29439914

SCH-50911 (162 words) [view diff] exact match in snippet view article find links to article

Sch 50911 and related compounds as novel GABAB antagonists". Bioorganic & Medicinal Chemistry Letters. 6 (13): 1529–34. doi:10.1016/S0960-894X(96)00267-3

5-HT2C receptor agonist (5,032 words) [view diff] exact match in snippet view article find links to article

highly selective 5HT2c agonists for the treatment of obesity". Bioorganic & Medicinal Chemistry Letters. 20 (7): 2365–9. doi:10.1016/j.bmcl.2010.01.107. PMID 20202843

Isoxazole (588 words) [view diff] exact match in snippet view article find links to article

"The recent progress of isoxazole in medicinal chemistry". Bioorganic & Medicinal Chemistry. 26 (12): 3065–3075. doi:10.1016/j.bmc.2018.05.013. Clemens

PD-102,807 (343 words) [view diff] exact match in snippet view article find links to article

"Diphenidol-related diamines as novel muscarinic M4 receptor antagonists". Bioorganic & Medicinal Chemistry Letters. 18 (9): 2972–6. doi:10.1016/j.bmcl.2008.03.061. PMID 18395442

Salinispora arenicola (221 words) [view diff] exact match in snippet view article find links to article

development of the anticancer agent salinosporamide A (NPI-0052)". Bioorganic & Medicinal Chemistry. 17 (6): 2175–2180. doi:10.1016/j.bmc.2008.10.075. PMC 2814440

Spongiacidin (87 words) [view diff] exact match in snippet view article find links to article

sponge Stylissa massa, functions as a USP7 inhibitor" (PDF). Bioorganic & Medicinal Chemistry Letters. 23 (13): 3884–6. doi:10.1016/j.bmcl.2013.04.066. PMID 23684893

Discovery and development of HIV-protease inhibitors (4,117 words) [view diff] exact match in snippet view article find links to article

containing novel dimethylphenoxyl acetates as P2 ligands". Bioorganic & Medicinal Chemistry Letters. 13 (21): 3657–60. doi:10.1016/j.bmcl.2003.08.043.

Bifonazole (486 words) [view diff] exact match in snippet view article find links to article

rigidification and influence of substituents at the methylene bridge". Bioorganic & Medicinal Chemistry. 16 (16): 7715–7727. doi:10.1016/j.bmc.2008.07.011. PMID 18674917

Calanolide A (2,249 words) [view diff] exact match in snippet view article find links to article

rainforest tree Calophyllum teysmannii var. inophylloide". Bioorganic & Medicinal Chemistry Letters. 4 (16): 1961–1964. doi:10.1016/S0960-894X(01)80543-6

Ganoderol A (92 words) [view diff] exact match in snippet view article find links to article

ganoderol B isolated from the fruiting body of Ganoderma lucidum". Bioorganic & Medicinal Chemistry. 15 (14): 4966–72. doi:10.1016/j.bmc.2007.04.036. PMID 17499997

Carbonic anhydrase 5A, mitochondrial (339 words) [view diff] exact match in snippet view article find links to article

mitochondrial isoforms VA and VB with amino acids and amines". Bioorganic & Medicinal Chemistry Letters. 17 (5): 1336–40. doi:10.1016/j.bmcl.2006.11.075. PMID 17174092

Xue-Min Cheng (793 words) [view diff] exact match in snippet view article find links to article

"Ketopiperazine-based renin inhibitors: Optimization of the "C" ring". Bioorganic & Medicinal Chemistry Letters. 16 (9): 2500–2504. doi:10.1016/j.bmcl.2006.01.084

Algaecide (528 words) [view diff] exact match in snippet view article find links to article

"Chemical reactivity and microbicidal action of bethoxazin". Bioorganic & Medicinal Chemistry. 20 (4): 1494–501. doi:10.1016/j.bmc.2011.12.051. PMID 22264763

AZD9272 (333 words) [view diff] exact match in snippet view article find links to article

allosteric modulators selected for clinical development". Bioorganic & Medicinal Chemistry Letters. 22 (22): 6974–6979. doi:10.1016/j.bmcl.2012.08.100

Carbonic anhydrase 7 (470 words) [view diff] exact match in snippet view article find links to article

isozyme VII with aromatic and heterocyclic sulfonamides". Bioorganic & Medicinal Chemistry Letters. 15 (4): 971–6. doi:10.1016/j.bmcl.2004.12.052. PMID 15686895

Discovery and development of NS5A inhibitors (5,211 words) [view diff] exact match in snippet view article find links to article

around the tetracyclic indole class of HCV NS5A inhibitors". Bioorganic & Medicinal Chemistry Letters. 26 (20): 5132–5137. doi:10.1016/j.bmcl.2016.07.057

Cannabigerovarin (535 words) [view diff] exact match in snippet view article find links to article

and its analogs: a review of their effects on inflammation". Bioorganic & Medicinal Chemistry. 23 (7): 1377–1385. doi:10.1016/j.bmc.2015.01.059. ISSN 0968-0896

Maslinic acid (572 words) [view diff] exact match in snippet view article find links to article

as a new class of inhibitors of glycogen phosphorylases". Bioorganic & Medicinal Chemistry Letters. 15 (22): 4944–4948. doi:10.1016/j.bmcl.2005.08.026

3,3-Diphenylpropylamine (87 words) [view diff] exact match in snippet view article find links to article

"Novel sterically hindered cannabinoid CB1 receptor ligands". Bioorganic & Medicinal Chemistry. 16 (15): 7510–7515. doi:10.1016/j.bmc.2008.06.001. hdl:11563/122572

5''-phosphoribostamycin phosphatase (99 words) [view diff] exact match in snippet view article find links to article

"Unique O-ribosylation in the biosynthesis of butirosin". Bioorganic & Medicinal Chemistry. 15 (13): 4360–8. doi:10.1016/j.bmc.2007.04.040. PMID 17482823

Balaram Mukhopadhyay (1,098 words) [view diff] exact match in snippet view article find links to article

Rajput, Hakon Leffler, Ulf J. Nilsson and Balaram Mukhopadhyay, Bioorganic & Medicinal Chemistry Letters 2014, 24, 3516–3520. Iodine monobromide - update. R

SB-705498 (295 words) [view diff] exact match in snippet view article find links to article

bioavailable TRPV1 antagonist suitable for clinical development". Bioorganic & Medicinal Chemistry Letters. 16 (12): 3287–91. doi:10.1016/j.bmcl.2006.03.030.

Fluorolintane (328 words) [view diff] exact match in snippet view article find links to article

2-diphenylethyl)piperidine enantiomers and of related compounds". Bioorganic & Medicinal Chemistry. 17 (9): 3456–62. doi:10.1016/j.bmc.2009.03.025. PMID 19345586

Discovery and development of NS5A inhibitors (5,211 words) [view diff] exact match in snippet view article find links to article

around the tetracyclic indole class of HCV NS5A inhibitors". Bioorganic & Medicinal Chemistry Letters. 26 (20): 5132–5137. doi:10.1016/j.bmcl.2016.07.057

Proteolysis targeting chimera (1,566 words) [view diff] exact match in snippet view article find links to article

induced by a small molecule: En route to chemical proteomics". Bioorganic & Medicinal Chemistry Letters. 18 (22): 5904–5908. doi:10.1016/j.bmcl.2008.07.114

JWH-007 (661 words) [view diff] exact match in snippet view article find links to article

"Design, Synthesis and Pharmacology of Cannabimimetic Indoles". Bioorganic & Medicinal Chemistry Letters. 4 (4): 563–566. doi:10.1016/s0960-894x(01)80155-4

RQ-00203078 (182 words) [view diff] exact match in snippet view article find links to article

RQ-00203078, as a selective and orally active TRPM8 antagonist". Bioorganic & Medicinal Chemistry Letters. 24 (23): 5364–8. doi:10.1016/j.bmcl.2014.10.074. PMID 25455182

RN-9893 (132 words) [view diff] exact match in snippet view article find links to article

orally-bioavailable antagonists of the TRPV4 ion-channel". Bioorganic & Medicinal Chemistry Letters. 25 (18): 4011–5. doi:10.1016/j.bmcl.2015.06.098. PMID 26235950

CXCR3 (2,039 words) [view diff] exact match in snippet view article find links to article

3: Tropenyl and homotropenyl-piperidine urea derivatives". Bioorganic & Medicinal Chemistry Letters. 18 (1): 147–151. doi:10.1016/j.bmcl.2007.10.109. PMID 18032038

Affinisine (301 words) [view diff] exact match in snippet view article find links to article

(Müell. Arg) Miers that inhibit acetylcholinesterase enzyme". Bioorganic & Medicinal Chemistry. 13 (12): 4092–4095. doi:10.1016/j.bmc.2005.03.045. PMID 15911323

S-Adenosyl-L-homocysteine (260 words) [view diff] exact match in snippet view article find links to article

methyltransferases by S-adenosyl-L-homocysteine analogues". Bioorganic & Medicinal Chemistry. 16 (5): 2276–2285. doi:10.1016/j.bmc.2007.11.075. PMID 18083524

Befetupitant (164 words) [view diff] exact match in snippet view article find links to article

selective, orally active neurokinin-1 receptor antagonists". Bioorganic & Medicinal Chemistry Letters. 16 (5): 1362–5. doi:10.1016/j.bmcl.2005.11.047. PMID 16332435

Thunberginol A (174 words) [view diff] exact match in snippet view article find links to article

folium on splenocyte proliferation activated by mitogens". Bioorganic & Medicinal Chemistry Letters. 8 (3): 215–20. doi:10.1016/S0960-894X(97)10221-9.

Flavonoid alkaloid (294 words) [view diff] exact match in snippet view article find links to article

of novel flavonoid alkaloids as α-glucosidase inhibitors. Bioorganic & Medicinal Chemistry. Jain SK, Bharate SB, Vishwakarma RA (2012). "Cyclin-dependent

Gabriel–Colman rearrangement (831 words) [view diff] exact match in snippet view article find links to article

of human leukocyte elastase, cathepsin G and proteinase 3". Bioorganic & Medicinal Chemistry. 3 (2): 187–193. doi:10.1016/0968-0896(95)00013-7. PMID 7796053

TCS-OX2-29 (154 words) [view diff] exact match in snippet view article find links to article

first orexin-2 receptor selective non-peptidic antagonist". Bioorganic & Medicinal Chemistry Letters. 13 (24): 4497–9. doi:10.1016/j.bmcl.2003.08.038. PMID 14643355

JWH-133 (598 words) [view diff] exact match in snippet view article find links to article

compounds: synthesis of selective ligands for the CB2 receptor". Bioorganic & Medicinal Chemistry. 7 (12): 2905–2914. doi:10.1016/S0968-0896(99)00219-9. PMID 10658595

3C-like protease (1,654 words) [view diff] exact match in snippet view article find links to article

mutant of SARS 3CL protease as a proteolysis-resistant mutant". Bioorganic & Medicinal Chemistry. 16 (21): 9400–8. doi:10.1016/j.bmc.2008.09.057. PMC 7126698

RTI-353 (146 words) [view diff] exact match in snippet view article find links to article

2beta-carbomethoxy-3beta-[aryl or heteroaryl]phenyltropanes". Bioorganic & Medicinal Chemistry Letters. 16 (1): 217–20. doi:10.1016/j.bmcl.2005.09.016. PMID 16236497

Eugeroic (1,928 words) [view diff] exact match in snippet view article find links to article

"Wake-promoting agents: search for next generation modafinil: part I". Bioorganic & Medicinal Chemistry Letters. 22 (6): 2312–2314. doi:10.1016/j.bmcl.2011.12.099

BHF-177 (136 words) [view diff] exact match in snippet view article find links to article

analogues as positive allosteric modulators of GABA B receptors". Bioorganic & Medicinal Chemistry Letters. 17 (22): 6206–11. doi:10.1016/j.bmcl.2007.09.023.

Adarotene (66 words) [view diff] exact match in snippet view article find links to article

(2012). "New retinoid derivatives as back-ups of Adarotene". Bioorganic & Medicinal Chemistry. 20 (7): 2405–15. doi:10.1016/j.bmc.2012.01.042. PMID 22365912

Discovery and development of integrase inhibitors (4,155 words) [view diff] exact match in snippet view article find links to article

scaffold hopping approach using salicylate and catechol groups". Bioorganic & Medicinal Chemistry. 19 (16): 4935–52. doi:10.1016/j.bmc.2011.06.058. PMC 3163123

Ibipinabant (547 words) [view diff] exact match in snippet view article find links to article

cannabinoid CB1 receptor antagonists with lower lipophilicity". Bioorganic & Medicinal Chemistry Letters. 15 (21): 4794–4798. doi:10.1016/j.bmcl.2005.07.054

Transphosphorylation (327 words) [view diff] exact match in snippet view article find links to article

ultra-high throughput screening against human and mouse isozymes". Bioorganic & Medicinal Chemistry Letters. 24 (3): 1000–1004. doi:10.1016/j.bmcl.2013.12.043

A-349821 (207 words) [view diff] exact match in snippet view article find links to article

novel and selective histamine H3 receptor antagonists". Bioorganic & Medicinal Chemistry Letters. 13 (7): 1325–8. doi:10.1016/S0960-894X(03)00118-5

Ligand efficiency (576 words) [view diff] exact match in snippet view article find links to article

Strengths and limitations of commonly used composite parameters". Bioorganic & Medicinal Chemistry Letters. 23 (21): 5980–5991. doi:10.1016/j.bmcl.2013.08.029

JD5037 (528 words) [view diff] exact match in snippet view article find links to article

metabolic disorder therapeutics devoid of CNS liabilities". Bioorganic & Medicinal Chemistry Letters. 22 (19): 6173–6180. doi:10.1016/j.bmcl.2012.08.004

WMS-2539 (62 words) [view diff] exact match in snippet view article find links to article

dexoxadrol analogues as uncompetitive NMDA receptor antagonists". Bioorganic & Medicinal Chemistry. 18 (22): 7855–7867. doi:10.1016/j.bmc.2010.09.047. PMID 20965735

Argyrochosma nivea (1,730 words) [view diff] exact match in snippet view article find links to article

system. A new skeletal basis for antiplasmodial compounds". Bioorganic & Medicinal Chemistry Letters. 13 (16): 2769–72. doi:10.1016/S0960-894X(03)00509-2

1-Amino-5-phosphonoindan-1-carboxylic acid (275 words) [view diff] exact match in snippet view article find links to article

and MCPG as metabotropic glutamate receptor antagonists". Bioorganic & Medicinal Chemistry Letters. 7 (9): 1195–1198. doi:10.1016/S0960-894X(97)00177-7

Neotripterifordin (76 words) [view diff] exact match in snippet view article find links to article

Tripterygium wilfordii: Isolation and structural elucidation". Bioorganic & Medicinal Chemistry. 3 (10): 1345–1348. doi:10.1016/0968-0896(95)00114-v. PMID 8564400

Serotonin transporter (3,438 words) [view diff] exact match in snippet view article find links to article

discovery of a selective SERT antagonist with picomolar potency". Bioorganic & Medicinal Chemistry Letters. 15 (4): 1131–1133. doi:10.1016/j.bmcl.2004.12.014

Totarol (5,462 words) [view diff] exact match in snippet view article find links to article

derivatives. Part 1: modifications of ring-C and pro-drugs". Bioorganic & Medicinal Chemistry. 7 (9): 1953–1964. doi:10.1016/s0968-0896(99)00162-5. PMID 10530944

Smallanthus fruticosus (122 words) [view diff] exact match in snippet view article find links to article

M. Lin, Ernest Hamel, Gordon M. Cragg and Michael R. Boyd, Bioorganic & Medicinal Chemistry Letters, Volume 3, Issue 4, April 1993, pages 581-584, doi:10

JNJ-28330835 (178 words) [view diff] exact match in snippet view article find links to article

imidazolopyrazole scaffold as selective androgen receptor modulators". Bioorganic & Medicinal Chemistry Letters. 17 (2): 439–43. doi:10.1016/j.bmcl.2006.10.035. PMID 17079140

Durantin A (56 words) [view diff] exact match in snippet view article find links to article

antioxidative coumarinolignoids from Duranta repens Linn". Bioorganic & Medicinal Chemistry Letters. 19 (13): 3521–3524. doi:10.1016/j.bmcl.2009.05.006

Cyclothiazomycin (1,132 words) [view diff] exact match in snippet view article find links to article

polymerase inhibitor, cyclothiazomycin B1, and its isomer". Bioorganic & Medicinal Chemistry. 14 (24): 8259–8270. doi:10.1016/j.bmc.2006.09.006. PMID 17010619

Nicotinic agonist (4,283 words) [view diff] exact match in snippet view article find links to article

SEN12333/WAY-317538: Novel alpha 7 nicotinic acetylcholine receptor agonist", Bioorganic & Medicinal Chemistry, 17 (14): 5247–5258, doi:10.1016/j.bmc.2009.05.040, PMID 19515567

Buprenorphine/samidorphan (1,992 words) [view diff] exact match in snippet view article find links to article

"Syntheses of novel high affinity ligands for opioid receptors". Bioorganic & Medicinal Chemistry Letters. 19 (8): 2289–2294. doi:10.1016/j.bmcl.2009.02.078

Christopher J. Schofield (4,203 words) [view diff] exact match in snippet view article find links to article

UK; Highly cited paper awards (e.g. Biochemical Journal, Bioorganic & Medicinal Chemistry Letters) 2009 – 2014: PI of ERC Advanced Investigator Grant

TC OT 39 (87 words) [view diff] exact match in snippet view article find links to article

Roe MB (September 2004). "Non-peptide oxytocin agonists". Bioorganic & Medicinal Chemistry Letters. 14 (17): 4585–4589. doi:10.1016/j.bmcl.2004.04.107

AFDX-384 (410 words) [view diff] exact match in snippet view article find links to article

AF-DX 384, a selective antagonist of muscarinic M2 receptors". Bioorganic & Medicinal Chemistry. 8 (3): 591–600. doi:10.1016/S0968-0896(99)00307-7. PMID 10732976

N-Methylornithine (127 words) [view diff] exact match in snippet view article find links to article

analogs as alternate substrates for nitric oxide synthase". Bioorganic & Medicinal Chemistry Letters. 15 (17): 3934–3941. doi:10.1016/j.bmcl.2005.05.088

Muscarinic acetylcholine receptor M5 (1,511 words) [view diff] exact match in snippet view article find links to article

"Discovery of ML326: The first sub-micromolar, selective M5 PAM". Bioorganic & Medicinal Chemistry Letters. 23 (10): 2996–3000. doi:10.1016/j.bmcl.2013.03.032

C286 (907 words) [view diff] exact match in snippet view article find links to article

and RAR β agonists as Orally Bioavailable Drugs. A review". Bioorganic & Medicinal Chemistry. 28 (20): 115664. doi:10.1016/j.bmc.2020.115664. PMC 7588594

Eleutherobin (76 words) [view diff] exact match in snippet view article find links to article

McCulloch, M. W; Kerr, R. G (2011). "Marine diterpene glycosides". Bioorganic & Medicinal Chemistry. 19 (22): 6702–19. doi:10.1016/j.bmc.2011.06.083. PMID 21783368

PD-168,077 (411 words) [view diff] exact match in snippet view article find links to article

selective dopamine D4 receptor agonists". Bioorganic & Medicinal Chemistry. 12 (13): 3471–3483. doi:10.1016/j.bmc.2004.04.035. PMID 15186832

PD-168,077 (411 words) [view diff] exact match in snippet view article find links to article

selective dopamine D4 receptor agonists". Bioorganic & Medicinal Chemistry. 12 (13): 3471–3483. doi:10.1016/j.bmc.2004.04.035. PMID 15186832

Xestoquinone (140 words) [view diff] exact match in snippet view article find links to article

inhibitor isolated from a Vanuatu marine sponge Xestospongia sp". Bioorganic & Medicinal Chemistry. 14 (13): 4477–4482. doi:10.1016/j.bmc.2006.02.026. ISSN 0968-0896

Aplysiatoxin (348 words) [view diff] exact match in snippet view article find links to article

simplified analogue of aplysiatoxin with antiproliferative activity. Bioorganic & Medicinal Chemistry Letters. 2010 Oct 15;20(20):6064-6. PMID 20817520

Eleutherobin (76 words) [view diff] exact match in snippet view article find links to article

McCulloch, M. W; Kerr, R. G (2011). "Marine diterpene glycosides". Bioorganic & Medicinal Chemistry. 19 (22): 6702–19. doi:10.1016/j.bmc.2011.06.083. PMID 21783368

Methylphenylpiracetam (536 words) [view diff] exact match in snippet view article find links to article

novel positive allosteric modulators of sigma-1 receptor". Bioorganic & Medicinal Chemistry. 21 (10): 2764–71. doi:10.1016/j.bmc.2013.03.016. PMID 23582449

3-Methoxymethamphetamine (144 words) [view diff] exact match in snippet view article find links to article

stereoselective binding site for compounds in the amphetamine class". Bioorganic & Medicinal Chemistry. 19 (23): 7044–7048. doi:10.1016/j.bmc.2011.10.007. PMC 3236098

Dihydro-resveratrol (224 words) [view diff] exact match in snippet view article find links to article

(2010). "Dihydro-resveratrol—A potent dietary polyphenol". Bioorganic & Medicinal Chemistry Letters. 20 (20): 6149–51. doi:10.1016/j.bmcl.2010.08.002.

Bergamottin (684 words) [view diff] exact match in snippet view article find links to article

and their effect on human CYP 3A4 and CYP 1B1 isoenzymes". Bioorganic & Medicinal Chemistry. 14 (8): 2606–2612. doi:10.1016/j.bmc.2005.11.039. PMID 16338240

PEAQX (175 words) [view diff] exact match in snippet view article find links to article

the human 1A/2A, rather than 1A/2B receptor composition". Bioorganic & Medicinal Chemistry Letters. 12 (7): 1099–102. doi:10.1016/s0960-894x(02)00074-4

Aldehyde oxidase (999 words) [view diff] exact match in snippet view article find links to article

chemistry approaches to avoid aldehyde oxidase metabolism". Bioorganic & Medicinal Chemistry Letters. 22 (8): 2856–60. doi:10.1016/j.bmcl.2012.02.069. PMID 22429467

Fluorodeoxyglycosylamine (315 words) [view diff] exact match in snippet view article find links to article

lipophilic amines for development of potential PET imaging agents". Bioorganic & Medicinal Chemistry Letters. 25 (15): 2902–2906. doi:10.1016/j.bmcl.2015.05.053

Zhankuic acid (203 words) [view diff] exact match in snippet view article find links to article

cell activation and the contact hypersensitivity response". Bioorganic & Medicinal Chemistry Letters. 25 (20): 4637–4641. doi:10.1016/j.bmcl.2015.08.038

Aurone (467 words) [view diff] exact match in snippet view article find links to article

(2017-02-15). "Antifungal activity of substituted aurones". Bioorganic & Medicinal Chemistry Letters. 27 (4): 901–903. doi:10.1016/j.bmcl.2017.01.012. PMID 28094180

4-Pyrone (222 words) [view diff] exact match in snippet view article find links to article

products—A privileged compound class provided by nature". Bioorganic & Medicinal Chemistry. 17 (6): 2304–2309. doi:10.1016/j.bmc.2008.11.001. PMID 19042133

Trifluralin (2,414 words) [view diff] exact match in snippet view article find links to article

evaluation of trifluralin analogues as antileishmanial agents". Bioorganic & Medicinal Chemistry. 18 (1): 274–281. doi:10.1016/j.bmc.2009.10.059. PMID 19926293

Karen Joy Shaw (2,518 words) [view diff] exact match in snippet view article find links to article

APX001A and in vitro evaluation against Cryptococcus spp. Bioorganic & Medicinal Chemistry Letters doi: https://doi.org/10.1016/j.bmcl. 2019.126713 Epub

Licochalcone A (258 words) [view diff] exact match in snippet view article find links to article

(H1N1) neuraminidase inhibitors from Glycyrrhiza inflata". Bioorganic & Medicinal Chemistry Letters. 21 (1): 294–8. doi:10.1016/j.bmcl.2010.11.016. PMID 21123068

Lisofylline (521 words) [view diff] exact match in snippet view article find links to article

(LSF) analogs as a potential treatment for Type 1 diabetes". Bioorganic & Medicinal Chemistry Letters. 16 (13): 3401–5. doi:10.1016/j.bmcl.2006.04.036. PMID 16650991

Azumolene (167 words) [view diff] exact match in snippet view article find links to article

Barreiro EJ (September 2018). "N-Acylhydrazones as drugs". Bioorganic & Medicinal Chemistry Letters. 28 (17): 2797–2806. doi:10.1016/j.bmcl.2018.07.015

Centaureidin (184 words) [view diff] exact match in snippet view article find links to article

from Polymnia fruticosa, inhibits tubulin polymerization". Bioorganic & Medicinal Chemistry Letters. 3 (4): 581–4. doi:10.1016/S0960-894X(01)81233-6. v

MGS-0039 (557 words) [view diff] exact match in snippet view article find links to article

group II mGluR antagonist with antidepressant-like potential". Bioorganic & Medicinal Chemistry. 14 (12): 4193–207. doi:10.1016/j.bmc.2006.01.060. PMID 16487713

3-Methyluridine (99 words) [view diff] exact match in snippet view article find links to article

RNA nucleosides: 3-methyluridine and 3-methylpseudouridine". Bioorganic & Medicinal Chemistry. 13 (24): 6777–6781. doi:10.1016/j.bmc.2005.07.061. ISSN 0968-0896

Salinosporamide (509 words) [view diff] exact match in snippet view article find links to article

development of the anticancer agent salinosporamide A (NPI-0052)". Bioorganic & Medicinal Chemistry. 17 (6): 2175–80. doi:10.1016/j.bmc.2008.10.075. PMC 2814440

Vindesine (197 words) [view diff] exact match in snippet view article find links to article

analogues as anti-cancer agents: Looking back, peering ahead". Bioorganic & Medicinal Chemistry Letters. 28 (17): 2816–2826. doi:10.1016/j.bmcl.2018.06.044

ATC-0175 (232 words) [view diff] exact match in snippet view article find links to article

antagonists for the melanin-concentrating hormone receptor 1". Bioorganic & Medicinal Chemistry Letters. 15 (17): 3853–6. doi:10.1016/j.bmcl.2005.05.121. PMID 16002290

Bruceolide (82 words) [view diff] exact match in snippet view article find links to article

"Anti-malarial activities of acylated bruceolide derivatives". Bioorganic & Medicinal Chemistry Letters. 8 (5): 459–462. doi:10.1016/S0960-894X(98)00045-6

PF-219,061 (270 words) [view diff] exact match in snippet view article find links to article

agonist and its in vivo delivery via the intranasal route". Bioorganic & Medicinal Chemistry Letters. 17 (24): 6691–6. doi:10.1016/j.bmcl.2007.10.059. PMID 17976986

Palmatine (2,153 words) [view diff] exact match in snippet view article find links to article

13-substituted palmatines and 8-oxo-13-substituted dihydropalmatines". Bioorganic & Medicinal Chemistry. 26 (9): 2586–2598. doi:10.1016/j.bmc.2018.04.025. ISSN 0968-0896

Stauprimide (174 words) [view diff] exact match in snippet view article find links to article

selectivity of staurosporine derivatives towards protein kinase C". Bioorganic & Medicinal Chemistry Letters. 4 (3): 399–404. doi:10.1016/0960-894X(94)80004-9.

17-Dimethylaminoethylamino-17-demethoxygeldanamycin (128 words) [view diff] exact match in snippet view article find links to article

"Structure-based design of 7-carbamate analogs of geldanamycin". Bioorganic & Medicinal Chemistry Letters. 15 (22): 5016–5021. doi:10.1016/j.bmcl.2005.08.013

6',7'-Dihydroxybergamottin (239 words) [view diff] exact match in snippet view article find links to article

and their effect on human CYP 3A4 and CYP 1B1 isoenzymes". Bioorganic & Medicinal Chemistry. 14 (8): 2606–2612. doi:10.1016/j.bmc.2005.11.039. ISSN 0968-0896

Chalcone (636 words) [view diff] exact match in snippet view article find links to article

2′-amino chalcones: design, synthesis and biological evaluation". Bioorganic & Medicinal Chemistry Letters. 10 (8): 699–701. doi:10.1016/S0960-894X(00)00072-X

Micromonospora lupini (266 words) [view diff] exact match in snippet view article find links to article

an endophytic actinomycete Micromonospora lupini sp. nov". Bioorganic & Medicinal Chemistry Letters. 17 (13): 3702–3705. doi:10.1016/j.bmcl.2007.04.039

DTDP-L-rhamnose 4-epimerase (132 words) [view diff] exact match in snippet view article find links to article

dTDP-L-rhamnose 4-epimerase in Burkholderia thailandensis". Bioorganic & Medicinal Chemistry Letters. 21 (13): 3914–7. doi:10.1016/j.bmcl.2011.05.030. PMID 21640586

Prodiamine (130 words) [view diff] exact match in snippet view article find links to article

evaluation of oryzalin analogs against Toxoplasma gondii". Bioorganic & Medicinal Chemistry Letters. 20 (17): 5179. doi:10.1016/j.bmcl.2010.07.003. PMC 2922421

Lambertella corni-maris (1,050 words) [view diff] exact match in snippet view article find links to article

and novel biosynthetic congener of lambertellols A and B". Bioorganic & Medicinal Chemistry Letters. 15 (10): 2587–2590. doi:10.1016/j.bmcl.2005.03.036

Lortalamine (368 words) [view diff] exact match in snippet view article find links to article

and oxaprotiline) for comparative PET studies in baboons". Bioorganic & Medicinal Chemistry. 13 (15): 4658–66. doi:10.1016/j.bmc.2005.04.062. PMID 15914010

5-HT2A receptor (9,998 words) [view diff] exact match in snippet view article find links to article

agonist 5-HT2A/2C receptor PET radioligand in nonhuman primate". Bioorganic & Medicinal Chemistry Letters. 27 (1): 21–23. doi:10.1016/j.bmcl.2016.11.043. PMC 5348621

Lobeline (1,249 words) [view diff] exact match in snippet view article find links to article

tetrabenazine analogs for the vesicular monoamine transporter-2". Bioorganic & Medicinal Chemistry. 15 (8): 2975–92. doi:10.1016/j.bmc.2007.02.013. PMC 2001191

Inte:Ligand (1,728 words) [view diff] exact match in snippet view article find links to article

silico exploration for agonists/antagonists of brassinolide". Bioorganic & Medicinal Chemistry Letters. 26 (7): 1709–1714. doi:10.1016/j.bmcl.2016.02.054

Sarmazenil (254 words) [view diff] exact match in snippet view article find links to article

(benzodiazepine receptors): comparison with bretazenil and flumazenil". Bioorganic & Medicinal Chemistry. 6 (10): 1745–57. doi:10.1016/S0968-0896(98)00117-5. PMID 9839004

Salvinorin B methoxymethyl ether (535 words) [view diff] exact match in snippet view article find links to article

pharmacological studies of new C(2) modified salvinorin A analogues". Bioorganic & Medicinal Chemistry Letters. 15 (16): 3744–3747. doi:10.1016/j.bmcl.2005.05.048

Novodinia antillensis (475 words) [view diff] exact match in snippet view article find links to article

Sch 725739, from a marine starfish, Novodinia antillensis". Bioorganic & Medicinal Chemistry Letters. 7 (20): 5543–5547. doi:10.1016/j.bmcl.2007.08.025

N6-Cyclopentyladenosine (352 words) [view diff] exact match in snippet view article find links to article

selective, high affinity adenosine A1 receptor agonists". Bioorganic & Medicinal Chemistry Letters. 17 (1): 161–166. doi:10.1016/j.bmcl.2006.09.065. PMID 17045477

Evocalcet (177 words) [view diff] exact match in snippet view article find links to article

receptor agonist for the treatment of hyperparathyroidism". Bioorganic & Medicinal Chemistry Letters. 28 (11): 2055–2060. doi:10.1016/j.bmcl.2018.04.055

Rhazinilam (155 words) [view diff] exact match in snippet view article find links to article

structure - activity relationships on tubulin-microtubule system". Bioorganic & Medicinal Chemistry Letters. 7 (17): 2155–2158. doi:10.1016/S0960-894X(97)00391-0

Baicalin (615 words) [view diff] exact match in snippet view article find links to article

able to reach the CNS, is a prolyl oligopeptidase inhibitor". Bioorganic & Medicinal Chemistry. 16 (15): 7516–24. doi:10.1016/j.bmc.2008.04.067. PMID 18650094

Ramoplanin (700 words) [view diff] exact match in snippet view article find links to article

biosynthesis of the lipodepsipeptide antibiotic Ramoplanin A2". Bioorganic & Medicinal Chemistry. 20 (2): 859–865. doi:10.1016/j.bmc.2011.11.062. PMID 22222159

PF-05089771 (198 words) [view diff] exact match in snippet view article find links to article

"Recent progress in sodium channel modulators for pain". Bioorganic & Medicinal Chemistry Letters. 24 (16): 3690–3699. doi:10.1016/j.bmcl.2014.06.038

Rhazinilam (155 words) [view diff] exact match in snippet view article find links to article

structure - activity relationships on tubulin-microtubule system". Bioorganic & Medicinal Chemistry Letters. 7 (17): 2155–2158. doi:10.1016/S0960-894X(97)00391-0

Yoshito Kishi (432 words) [view diff] exact match in snippet view article find links to article

"Tetrahedron Prize for Creativity in Organic Chemistry or Bioorganic & Medicinal Chemistry". Elsevier. Archived from the original on September 9, 2014

Methylpiperidinopyrazole (170 words) [view diff] exact match in snippet view article find links to article

antiestrogens with estrogen receptor alpha selective activity". Bioorganic & Medicinal Chemistry Letters. 19 (1): 108–10. doi:10.1016/j.bmcl.2008.11.006. PMC 2711511

PF-05089771 (198 words) [view diff] exact match in snippet view article find links to article

"Recent progress in sodium channel modulators for pain". Bioorganic & Medicinal Chemistry Letters. 24 (16): 3690–3699. doi:10.1016/j.bmcl.2014.06.038

Desformylflustrabromine (829 words) [view diff] exact match in snippet view article find links to article

evaluation as an alpha4beta2 and alpha7 nACh receptor modulator". Bioorganic & Medicinal Chemistry Letters. 17 (17): 4855–4860. doi:10.1016/j.bmcl.2007.06.047

Dichroa febrifuga (467 words) [view diff] exact match in snippet view article find links to article

of febrifugine analogues as potential antimalarial agents". Bioorganic & Medicinal Chemistry Letters. 16 (7): 1854–1858. doi:10.1016/j.bmcl.2006.01.009

Seletracetam (2,338 words) [view diff] exact match in snippet view article find links to article

to find new anticonvulsant drugs from chemical diversity". Bioorganic & Medicinal Chemistry Letters. 13 (16): 2749–2754. doi:10.1016/S0960-894X(03)00535-3

Salinispora tropica (390 words) [view diff] exact match in snippet view article find links to article

development of the anticancer agent salinosporamide A (NPI-0052)". Bioorganic & Medicinal Chemistry. 17 (6): 2175–2180. doi:10.1016/j.bmc.2008.10.075. PMC 2814440

Neomycin (2,085 words) [view diff] exact match in snippet view article find links to article

"Unique O-ribosylation in the biosynthesis of butirosin". Bioorganic & Medicinal Chemistry. 15 (13): 4360–8. doi:10.1016/j.bmc.2007.04.040. PMID 17482823

Ro4938581 (318 words) [view diff] exact match in snippet view article find links to article

inverse agonists for the treatment of cognitive dysfunction". Bioorganic & Medicinal Chemistry Letters. 19 (20): 5940–4. doi:10.1016/j.bmcl.2009.08.053. PMID 19762240

RTIOX-276 (202 words) [view diff] exact match in snippet view article find links to article

tetrahydroisoquinolines as selective antagonists for the orexin 1 receptor". Bioorganic & Medicinal Chemistry. 23 (17): 5709–24. doi:10.1016/j.bmc.2015.07.013. PMC 4554834

UB-165 (354 words) [view diff] exact match in snippet view article find links to article

Identifying factors associated with alpha7 selectivity". Bioorganic & Medicinal Chemistry Letters. 13 (17): 2825–8. doi:10.1016/S0960-894X(03)00594-8

Dryopteris crassirhizoma (234 words) [view diff] exact match in snippet view article find links to article

acylphloroglucinols isolated from Dryopteris crassirhizoma". Bioorganic & Medicinal Chemistry Letters. 16 (18): 4738–42. doi:10.1016/j.bmcl.2006.07.018.

Antimetabolite (1,314 words) [view diff] exact match in snippet view article find links to article

from supramolecular principles to biological properties". Bioorganic & Medicinal Chemistry. 10 (4): 841–854. doi:10.1016/S0968-0896(01)00348-0. PMID 11836090

DAA-1097 (168 words) [view diff] exact match in snippet view article find links to article

derivatives as novel peripheral benzodiazepine receptor ligands". Bioorganic & Medicinal Chemistry. 12 (2): 423–38. doi:10.1016/j.bmc.2003.10.050. PMID 14723961

Metabotropic glutamate receptor 5 (3,032 words) [view diff] exact match in snippet view article find links to article

mGluR5 positive allosteric modulators: the discovery of CPPHA". Bioorganic & Medicinal Chemistry Letters. 17 (5): 1386–91. doi:10.1016/j.bmcl.2006.11.081. PMID 17210250

Ecklonia stolonifera (604 words) [view diff] exact match in snippet view article find links to article

isolated from Ecklonia stolonifera on Fc(epsilon)RI expression". Bioorganic & Medicinal Chemistry. 17 (13): 4734–9. doi:10.1016/j.bmc.2009.04.050. PMID 19443227

Iminocoumarin (481 words) [view diff] exact match in snippet view article find links to article

derivatives as potent inhibitors of tyrosine kinase p60c-src". Bioorganic & Medicinal Chemistry Letters. 5 (20). Elsevier BV: 2423–2428. doi:10.1016/0960-894x(95)00422-p

Sarcodon cyrneus (215 words) [view diff] exact match in snippet view article find links to article

activities of neurite genesis and nerve growth factor production". Bioorganic & Medicinal Chemistry. 15 (8): 2878–2882. doi:10.1016/j.bmc.2007.02.019. PMID 17320402

Diquafosol (120 words) [view diff] exact match in snippet view article find links to article

activity of a series of uridine dinucleoside 5'-polyphosphates". Bioorganic & Medicinal Chemistry Letters. 11 (2): 157–60. doi:10.1016/S0960-894X(00)00612-0

Funapide (239 words) [view diff] exact match in snippet view article find links to article

"Recent progress in sodium channel modulators for pain". Bioorganic & Medicinal Chemistry Letters. 24 (16): 3690–3699. doi:10.1016/j.bmcl.2014.06.038

BU09059 (182 words) [view diff] exact match in snippet view article find links to article

E (May 2014). "Antagonists of the kappa opioid receptor". Bioorganic & Medicinal Chemistry Letters. 24 (9): 2021–32. doi:10.1016/j.bmcl.2014.03.040. PMID 24690494

Distamycin (437 words) [view diff] exact match in snippet view article find links to article

between distamycin a and active moieties of antitumor agents". Bioorganic & Medicinal Chemistry. 15 (1): 17–35. doi:10.1016/j.bmc.2006.07.004. PMID 17081759

Sigma-1 receptor (3,052 words) [view diff] exact match in snippet view article find links to article

structure-affinity relationships and in vitro metabolic stability". Bioorganic & Medicinal Chemistry. 17 (10): 3630–3641. doi:10.1016/j.bmc.2009.03.060. PMID 19394833

Meshimakobu (1,007 words) [view diff] exact match in snippet view article find links to article

reductase produced by the medicinal fungus Phellinus linteus". Bioorganic & Medicinal Chemistry Letters. 21 (6): 1716–8. doi:10.1016/j.bmcl.2011.01.080. PMID 21316961

Cis,cis-1,3,5-Triaminocyclohexane (190 words) [view diff] exact match in snippet view article find links to article

derivatives for the preparation of gallium radiopharmaceuticals". Bioorganic & Medicinal Chemistry Letters. 6 (7): 807–810. doi:10.1016/0960-894X(96)00110-2.

2-Quinolone (200 words) [view diff] exact match in snippet view article find links to article

use of carbostyril in physiologically active substances". Bioorganic & Medicinal Chemistry Letters. 25 (17): 3415–3419. doi:10.1016/j.bmcl.2015.06.027

Serotonin–norepinephrine–dopamine reuptake inhibitor (15,840 words) [view diff] exact match in snippet view article find links to article

antagonist with high affinity for NK1 and NK2 receptors". Bioorganic & Medicinal Chemistry Letters. 6 (8): 951–6. doi:10.1016/0960-894X(96)00148-5. Xavier

Voacamine (237 words) [view diff] exact match in snippet view article find links to article

alkaloids with cannabinoid CB1 receptor antagonistic activity". Bioorganic & Medicinal Chemistry Letters. 21 (7): 1962–4. doi:10.1016/j.bmcl.2011.02.036. PMID 21376588

2C-B-BUTTERFLY (480 words) [view diff] exact match in snippet view article find links to article

"Substituted hexahydrobenzodipyrans as 5-HT2A/2C receptor probes". Bioorganic & Medicinal Chemistry. 10 (10): 3301–6. doi:10.1016/S0968-0896(02)00209-2. PMID 12150876

1,2,4-Triazole (560 words) [view diff] exact match in snippet view article find links to article

"The biology and chemistry of antifungal agents: A review". Bioorganic & Medicinal Chemistry. 20 (19): 5678–5698. doi:10.1016/j.bmc.2012.04.045. PMID 22902032

Huprine X (554 words) [view diff] exact match in snippet view article find links to article

Huprine derivatives as human acetylcholinesterase inhibitors". Bioorganic & Medicinal Chemistry. 17 (13): 4523–36. doi:10.1016/j.bmc.2009.05.005. PMID 19473849

Lacosamide (3,797 words) [view diff] exact match in snippet view article find links to article

pharmacological evaluation of conformationally restricted analogues". Bioorganic & Medicinal Chemistry. 9 (10): 2693–2708. doi:10.1016/s0968-0896(01)00204-8. PMID 11557357

DSP-2230 (122 words) [view diff] exact match in snippet view article find links to article

"Recent progress in sodium channel modulators for pain". Bioorganic & Medicinal Chemistry Letters. 24 (16): 3690–9. doi:10.1016/j.bmcl.2014.06.038. PMID 25060923

SRX246 (304 words) [view diff] exact match in snippet view article find links to article

(March 2007). "Azetidinones as vasopressin V1a antagonists". Bioorganic & Medicinal Chemistry. 15 (5): 2054–80. doi:10.1016/j.bmc.2006.12.031. PMC 2067992

Himeic acid A (64 words) [view diff] exact match in snippet view article find links to article

inhibitor isolated from a marine-derived fungus, Aspergillus sp". Bioorganic & Medicinal Chemistry Letters. 15 (1): 191–194. doi:10.1016/j.bmcl.2004.10.012. PMID 15582438

Odanacatib (274 words) [view diff] exact match in snippet view article find links to article

odanacatib (MK-0822), a selective inhibitor of cathepsin K". Bioorganic & Medicinal Chemistry Letters. 18 (3): 923–928. doi:10.1016/j.bmcl.2007.12.047. PMID 18226527

Borinic acid (1,880 words) [view diff] exact match in snippet view article find links to article

"Diphenylborinic acid is a strong inhibitor of serine proteases". Bioorganic & Medicinal Chemistry Letters. 4 (20): 2417–2420. doi:10.1016/S0960-894X(01)80401-7

AMG-517 (466 words) [view diff] exact match in snippet view article find links to article

vanilloid 1 (TRPV1) antagonists with improved solubility". Bioorganic & Medicinal Chemistry Letters. 17 (23): 6539–45. doi:10.1016/j.bmcl.2007.09.080.

Michellamine (365 words) [view diff] exact match in snippet view article find links to article

the tetrahydroisoquinoline rings for biological activity". Bioorganic & Medicinal Chemistry Letters. 7 (20): 2687–2690. doi:10.1016/S0960-894X(97)10057-9

NNC 45-0095 (279 words) [view diff] exact match in snippet view article find links to article

affinity non-steroidal agonist for the estrogen receptor". Bioorganic & Medicinal Chemistry Letters. 10 (4): 399–402. doi:10.1016/S0960-894X(00)00015-9

4-Methylmethylphenidate (454 words) [view diff] exact match in snippet view article find links to article

binding affinities at dopamine and serotonin transport sites". Bioorganic & Medicinal Chemistry Letters. 14 (7): 1799–802. doi:10.1016/j.bmcl.2003.12.097.

Estradiol sulfamate (1,643 words) [view diff] exact match in snippet view article find links to article

improved oral absorption and reduced hepatic interaction". Bioorganic & Medicinal Chemistry. 25 (20): 5569–5575. doi:10.1016/j.bmc.2017.08.027. PMID 28886996

L-741,626 (568 words) [view diff] exact match in snippet view article find links to article

receptor antagonist L741,626: Binding, function, and SAR". Bioorganic & Medicinal Chemistry Letters. 17 (3): 745–9. doi:10.1016/j.bmcl.2006.10.076. PMC 1851912

Norzoanthamine (194 words) [view diff] exact match in snippet view article find links to article

zoanthamine-type alkaloids on the aggregation of human platelets". Bioorganic & Medicinal Chemistry. 11 (10): 2301–2306. doi:10.1016/S0968-0896(03)00107-X. Miyashita

Mannopeptimycin glycopeptide (60 words) [view diff] exact match in snippet view article find links to article

ether derivatives of mannopeptimycin glycopeptide antibiotic". Bioorganic & Medicinal Chemistry Letters. 13 (6): 1151–1155. doi:10.1016/s0960-894x(03)00045-3

Derek Lowe (chemist) (829 words) [view diff] exact match in snippet view article

(5-(2H)-isoxazolonyl) ureas, potent inhibitors of hormone-sensitive lipase". Bioorganic & Medicinal Chemistry Letters. 14 (12): 3155–9. doi:10.1016/j.bmcl.2004.04.015. PMID 15149665

Protide (1,362 words) [view diff] exact match in snippet view article find links to article

replication in cells where the nucleoside is poorly active". Bioorganic & Medicinal Chemistry Letters. 2 (7): 701–704. doi:10.1016/S0960-894X(00)80395-9

H. V. Thulasiram (638 words) [view diff] exact match in snippet view article find links to article

enzymatic synthesis of antimicrobial andrographolide derivatives". Bioorganic & Medicinal Chemistry Letters. 28 (6): 1132–1137. doi:10.1016/j.bmcl.2018.01.007

List of miscellaneous 5HT2A agonists (1,928 words) [view diff] exact match in snippet view article find links to article

4]diazepino[1,7-a]indoles: new templates for 5-HT(2C) agonists". Bioorganic & Medicinal Chemistry Letters. 13 (14): 2369–2372. doi:10.1016/s0960-894x(03)00403-7

Repenin (172 words) [view diff] exact match in snippet view article find links to article

antioxidative coumarinolignoids from Duranta repens Linn". Bioorganic & Medicinal Chemistry Letters. 19 (13): 3521–3524. doi:10.1016/j.bmcl.2009.05.006

Phenylahistin (249 words) [view diff] exact match in snippet view article find links to article

mammalian cell cycle inhibitor produced by aspergillus ustus". Bioorganic & Medicinal Chemistry Letters. 7 (22): 2847–2852. doi:10.1016/S0960-894X(97)10104-4

Octahydroxyanthraquinone (201 words) [view diff] exact match in snippet view article find links to article

R (1995). "Hydroxy-anthraquinones as antimalarial agents". Bioorganic & Medicinal Chemistry Letters. 5 (17): 1927–1932. doi:10.1016/0960-894X(95)00326-O

Erythrina velutina (729 words) [view diff] exact match in snippet view article find links to article

alkaloid from Erythrina velutina, induced sleep on normal mice". Bioorganic & Medicinal Chemistry Letters. 18 (14): 3992–3994. doi:10.1016/j.bmcl.2008.06.002

Forasartan (943 words) [view diff] exact match in snippet view article find links to article

1 (AT1) selective nonpeptidic antagonists--a perspective". Bioorganic & Medicinal Chemistry. 18 (24): 8418–8456. doi:10.1016/j.bmc.2010.10.043. PMID 21071232

Salbostatin (182 words) [view diff] exact match in snippet view article find links to article

1995). "Total synthesis of trehalase inhibitor salbostatin". Bioorganic & Medicinal Chemistry Letters. 5 (5): 487–490. doi:10.1016/0960-894X(95)00055-X.

NK1 receptor antagonist (3,286 words) [view diff] exact match in snippet view article find links to article

selective, orally active neurokinin-1 receptor antagonists", Bioorganic & Medicinal Chemistry Letters, 16 (5): 1362–5, doi:10.1016/j.bmcl.2005.11.047, PMID 16332435

Ganoderic acid (299 words) [view diff] exact match in snippet view article find links to article

5α-reductase by triterpenoids isolated from Ganoderma lucidum". Bioorganic & Medicinal Chemistry. 14 (24): 8654–8660. doi:10.1016/j.bmc.2006.08.018. PMID 16962782

Talarozole (322 words) [view diff] exact match in snippet view article find links to article

3-[4-(arylamino)phenyl]-3-(azole)-2,2-dimethylpropanoates". Bioorganic & Medicinal Chemistry. 20 (20): 6080–6088. doi:10.1016/j.bmc.2012.08.044. PMID 22989911

Dopamine receptor D3 (3,180 words) [view diff] exact match in snippet view article find links to article

improvements of affinity and selectivity for D3 versus D2 receptors". Bioorganic & Medicinal Chemistry Letters. 19 (8): 2133–2138. doi:10.1016/j.bmcl.2009.03.015

Atagabalin (249 words) [view diff] exact match in snippet view article find links to article

"Synthesis and in vivo evaluation of bicyclic gababutins". Bioorganic & Medicinal Chemistry Letters. 20 (2): 461–4. doi:10.1016/j.bmcl.2009.11.118. PMID 20005103

EICAR (antiviral) (705 words) [view diff] exact match in snippet view article

imidazole nucleosides as potential anti-dengue virus agents". Bioorganic & Medicinal Chemistry. 27 (11): 2181–2186. doi:10.1016/j.bmc.2019.04.015. PMID 31003866

Verrulactone (66 words) [view diff] exact match in snippet view article find links to article

enoyl-ACP reductase produced by Penicillium verruculosum F375". Bioorganic & Medicinal Chemistry Letters. 22 (7): 2503–6. doi:10.1016/j.bmcl.2012.02.001. PMID 22377515

AM-855 (118 words) [view diff] exact match in snippet view article find links to article

restricted tetracyclic analogs of Δ8-tetrahydrocannabinol". Bioorganic & Medicinal Chemistry Letters. 9 (15): 2119–24. doi:10.1016/S0960-894X(99)00355-8

Purpurogallin (351 words) [view diff] exact match in snippet view article find links to article

estradiol methylation: Kinetics and in silico modeling studies". Bioorganic & Medicinal Chemistry. 13 (7): 2501–7. doi:10.1016/j.bmc.2005.01.037. PMID 15755652

CD38 (3,825 words) [view diff] exact match in snippet view article find links to article

Muller-Steffner H (July 2011). "Flavonoids as inhibitors of human CD38". Bioorganic & Medicinal Chemistry Letters. 21 (13): 3939–42. doi:10.1016/j.bmcl.2011.05.022.

JWH-184 (136 words) [view diff] exact match in snippet view article find links to article

stacking interactions with the CB(1) cannabinoid receptor". Bioorganic & Medicinal Chemistry. 11 (4): 539–49. doi:10.1016/s0968-0896(02)00451-0. PMID 12538019

GS-39783 (590 words) [view diff] exact match in snippet view article find links to article

analogues as positive allosteric modulators of GABA B receptors". Bioorganic & Medicinal Chemistry Letters. 17 (22): 6206–11. doi:10.1016/j.bmcl.2007.09.023.

JWH-116 (135 words) [view diff] exact match in snippet view article find links to article

stacking interactions with the CB(1) cannabinoid receptor". Bioorganic & Medicinal Chemistry. 11 (4): 539–49. doi:10.1016/s0968-0896(02)00451-0. PMID 12538019

Neuropeptide S (1,144 words) [view diff] exact match in snippet view article find links to article

"Structure-activity study at positions 3 and 4 of human neuropeptide S". Bioorganic & Medicinal Chemistry. 16 (19): 8841–5. doi:10.1016/j.bmc.2008.08.073. PMID 18793857

WAY-629 (69 words) [view diff] exact match in snippet view article find links to article

4]benzodiazepinoindoles are agonists at the human 5-HT2C receptor". Bioorganic & Medicinal Chemistry Letters. 14 (10): 2603–7. doi:10.1016/j.bmcl.2004.02.100. PMID 15109661

Intrinsic activity (973 words) [view diff] exact match in snippet view article find links to article

conditionally-silent agonist for the α7 nicotinic acetylcholine receptor". Bioorganic & Medicinal Chemistry Letters. 23 (14): 4145–4149. doi:10.1016/j.bmcl.2013.05.039

A-84,543 (267 words) [view diff] exact match in snippet view article find links to article

A-84543, a potent nicotinic acetylcholine receptor agonist". Bioorganic & Medicinal Chemistry Letters. 8 (3): 249–54. doi:10.1016/S0960-894X(98)00019-5.

Murepavadin (1,186 words) [view diff] exact match in snippet view article find links to article

based on the cationic antimicrobial peptide protegrin I". Bioorganic & Medicinal Chemistry. 13 (6): 2055–2064. doi:10.1016/j.bmc.2005.01.009. PMID 15727859

Pinoresinol (863 words) [view diff] exact match in snippet view article find links to article

(Sesamum indicum) seeds though inhibiting α-glucosidase". Bioorganic & Medicinal Chemistry Letters. 22 (16): 5215–7. doi:10.1016/j.bmcl.2012.06.068. PMID 22818971

Deekonda2016 (251 words) [view diff] exact match in snippet view article find links to article

derivatives as potent opioid receptor ligands". Bioorganic & Medicinal Chemistry. 23 (18): 6185–6194. doi:10.1016/j.bmc.2015.07.071. PMC 4642887

Curculigo orchioides (620 words) [view diff] exact match in snippet view article find links to article

(2008). "New polyphenols active on β-amyloid aggregation". Bioorganic & Medicinal Chemistry Letters. 18 (2): 828–831. doi:10.1016/j.bmcl.2007.11.028. PMID 18042380

Sorbinil (273 words) [view diff] exact match in snippet view article find links to article

active as aldose reductase inhibitors". Bioorganic & Medicinal Chemistry Letters. 21 (1): 200–3. doi:10.1016/j.bmcl.2010.11.041. PMID 21129963

Gosogliptin (720 words) [view diff] exact match in snippet view article find links to article

selective, orally active dipeptidyl peptidase IV inhibitor". Bioorganic & Medicinal Chemistry Letters. 19 (7): 1991–1995. doi:10.1016/j.bmcl.2009.02.041

RU-58841 (533 words) [view diff] exact match in snippet view article find links to article

arylhydantoins for investigation as androgen receptor radioligands". Bioorganic & Medicinal Chemistry Letters. 11 (8): 1045–1047. doi:10.1016/s0960-894x(01)00146-9

RecA (1,428 words) [view diff] exact match in snippet view article find links to article

"Directed molecular screening for RecA ATPase inhibitors". Bioorganic & Medicinal Chemistry Letters. 17 (12): 3249–3253. doi:10.1016/j.bmcl.2007.04.013

Pyrazole (1,143 words) [view diff] exact match in snippet view article find links to article

"Recently reported biological activities of pyrazole compounds". Bioorganic & Medicinal Chemistry. 25 (21): 5891–5903. doi:10.1016/j.bmc.2017.09.035. ISSN 0968-0896

Norbormide (3,264 words) [view diff] exact match in snippet view article find links to article

studies of analogues of the rat selective toxicant norbormide". Bioorganic & Medicinal Chemistry. 15 (8): 2963–74. doi:10.1016/j.bmc.2007.02.012. PMID 17321141

Brilanestrant (549 words) [view diff] exact match in snippet view article find links to article

regression in a tamoxifen-resistant breast cancer xenograft". Bioorganic & Medicinal Chemistry Letters. 25 (22): 5163–7. doi:10.1016/j.bmcl.2015.09.074. PMID 26463130

4-Nonylphenylboronic acid (154 words) [view diff] exact match in snippet view article find links to article

synthesis of boronic acid inhibitors of endothelial lipase". Bioorganic & Medicinal Chemistry Letters. 22 (3): 1397–401. doi:10.1016/j.bmcl.2011.12.043.

Hispidin (279 words) [view diff] exact match in snippet view article find links to article

antioxidants in the medicinal mushrooms Inonotus and Phellinus". Bioorganic & Medicinal Chemistry. 15 (10): 3309–14. doi:10.1016/j.bmc.2007.03.039. PMID 17387019

Hexaprenyl-diphosphate synthase ((2E,6E)-farnesyl-diphosphate specific) (231 words) [view diff] exact match in snippet view article

enzymes, hexaprenyl- and heptaprenyl diphosphate synthases". Bioorganic & Medicinal Chemistry Letters. 11 (16): 2157–9. doi:10.1016/S0960-894X(01)00391-2

Stylissa massa (246 words) [view diff] exact match in snippet view article find links to article

sponge Stylissa massa, functions as a USP7 inhibitor" (PDF). Bioorganic & Medicinal Chemistry Letters. 23 (13): 3884–6. doi:10.1016/j.bmcl.2013.04.066. PMID 23684893

CL-218,872 (462 words) [view diff] exact match in snippet view article find links to article

6-aryltriazolo-[4,3-b]pyridazine ligands of the benzodiazepine receptor". Bioorganic & Medicinal Chemistry. 2 (8): 773–9. doi:10.1016/s0968-0896(00)82176-8. PMID 7894970

3-Chloropropanoic acid (319 words) [view diff] exact match in snippet view article find links to article

gamma-hydroxybutyric acid receptor lacking a 4-hydroxyl group". Bioorganic & Medicinal Chemistry. 12 (7): 1643–1647. doi:10.1016/j.bmc.2004.01.025. PMID 15028257

Epibatidine (2,694 words) [view diff] exact match in snippet view article find links to article

affinity at neuronal nicotinic acetylcholine receptor subtypes". Bioorganic & Medicinal Chemistry Letters. 18 (16): 4651–4654. doi:10.1016/j.bmcl.2008.07.016

Miquelianin (435 words) [view diff] exact match in snippet view article find links to article

and structure–activity correlations with related alkaloids". Bioorganic & Medicinal Chemistry. 13 (2): 443–448. doi:10.1016/j.bmc.2004.10.020. PMID 15598565

SN-22 (332 words) [view diff] exact match in snippet view article find links to article

derivatives are potent and selective 5-HT6 receptor antagonists". Bioorganic & Medicinal Chemistry Letters. 15 (2): 379–83. doi:10.1016/j.bmcl.2004.10.064. PMID 15603958

ZD6126 (221 words) [view diff] exact match in snippet view article find links to article

Lippert JW (January 2007). "Vascular disrupting agents". Bioorganic & Medicinal Chemistry. 15 (2): 605–15. doi:10.1016/j.bmc.2006.10.020. PMID 17070061

Neuropeptide Y receptor Y5 (997 words) [view diff] exact match in snippet view article find links to article

and selective small molecule NPY Y5 receptor antagonists". Bioorganic & Medicinal Chemistry Letters. 12 (13): 1767–9. doi:10.1016/S0960-894X(02)00287-1

Cryptophycin (893 words) [view diff] exact match in snippet view article find links to article

mitotic and interphase impairment of microtubule function". Bioorganic & Medicinal Chemistry. 22 (18): 5050–5059. doi:10.1016/j.bmc.2014.02.035. PMID 24650703

SM-130686 (333 words) [view diff] exact match in snippet view article find links to article

relationships of the oxindole growth hormone secretagogues". Bioorganic & Medicinal Chemistry Letters. 15 (7): 1789–92. doi:10.1016/j.bmcl.2005.02.042. PMID 15780607

SN-22 (332 words) [view diff] exact match in snippet view article find links to article

derivatives are potent and selective 5-HT6 receptor antagonists". Bioorganic & Medicinal Chemistry Letters. 15 (2): 379–83. doi:10.1016/j.bmcl.2004.10.064. PMID 15603958

Neuraminidase inhibitor (1,048 words) [view diff] exact match in snippet view article find links to article

isoquinoline alkaloids from Corydalis turtschaninovii rhizome". Bioorganic & Medicinal Chemistry. 22 (21): 6047–6052. doi:10.1016/j.bmc.2014.09.004. PMID 25277281

Vimseltinib (92 words) [view diff] exact match in snippet view article find links to article

for the treatment of Tenosynovial Giant Cell Tumor (TGCT)". Bioorganic & Medicinal Chemistry Letters. 74: 128928. doi:10.1016/j.bmcl.2022.128928. PMID 35961460

Interfungin (78 words) [view diff] exact match in snippet view article find links to article

NF-κB inhibitory effects from the fungus Phellinus baumii". Bioorganic & Medicinal Chemistry Letters. 21 (11): 3261–7. doi:10.1016/j.bmcl.2011.04.025. PMID 21531558

AMG-41 (189 words) [view diff] exact match in snippet view article find links to article

"Novel 1',1'-chain substituted Delta(8)-tetrahydrocannabinols". Bioorganic & Medicinal Chemistry Letters. 12 (24): 3583–6. doi:10.1016/s0960-894x(02)00785-0

3-Bromomethylphenidate (188 words) [view diff] exact match in snippet view article find links to article

structure-activity relationship studies of threo-methylphenidate analogs". Bioorganic & Medicinal Chemistry. 18 (20): 7221–38. doi:10.1016/j.bmc.2010.08.034. PMID 20846865

Zosuquidar (592 words) [view diff] exact match in snippet view article find links to article

as potent multidrug resistance reversal agents". Bioorganic & Medicinal Chemistry Letters 5 (21): 2473–2476. doi:10.1016/0960-894X(95)00426-T

LASSBio-881 (179 words) [view diff] exact match in snippet view article find links to article

Discovery of LASSBio-881, a new ligand of cannabinoid receptors". Bioorganic & Medicinal Chemistry. 15 (6): 2421–33. doi:10.1016/j.bmc.2007.01.013. PMID 17275312

Iclaprim (1,069 words) [view diff] exact match in snippet view article find links to article

activity on trimethoprim sensitive and resistant bacteria". Bioorganic & Medicinal Chemistry Letters. 13 (23): 4217–4221. doi:10.1016/j.bmcl.2003.07.023

Cilomilast (492 words) [view diff] exact match in snippet view article find links to article

"Highly potent PDE4 inhibitors with therapeutic potential". Bioorganic & Medicinal Chemistry Letters. 14 (1): 207–10. doi:10.1016/j.bmcl.2003.09.087. PMID 14684329

Avermectin (1,799 words) [view diff] exact match in snippet view article find links to article

Hans (2009). "New ventures in the chemistry of avermectins". Bioorganic & Medicinal Chemistry. 17 (12): 4085–4095. doi:10.1016/j.bmc.2008.12.069. PMID 19168364

Tolimidone (472 words) [view diff] exact match in snippet view article find links to article

novel Lyn kinase activator with clinical proof of concept". Bioorganic & Medicinal Chemistry. 28 (9): 115425. doi:10.1016/j.bmc.2020.115425. PMID 32201192

Lomerizine (1,470 words) [view diff] exact match in snippet view article find links to article

as selective analgesic N-type calcium channel blockers". Bioorganic & Medicinal Chemistry Letters. 17 (3): 662–667. doi:10.1016/j.bmcl.2006.10.098. PMID 17134896

Thuja standishii (332 words) [view diff] exact match in snippet view article find links to article

structure–activity relationship of inhibitory activity against aromatase". Bioorganic & Medicinal Chemistry. 15 (7): 2736–2748. doi:10.1016/j.bmc.2007.01.031. PMID 17287126

Epristeride (992 words) [view diff] exact match in snippet view article find links to article

5(6)-steroids as new potential 5 alpha-reductase inhibitor". Bioorganic & Medicinal Chemistry Letters. 8 (15): 1949–1952. doi:10.1016/S0960-894X(98)00339-4

Allyl isothiocyanate (846 words) [view diff] exact match in snippet view article find links to article

Non-Electrophilic Reference Agonist of the TrpA1 Channel". Bioorganic & Medicinal Chemistry Letters. 21 (16): 4857–4859. doi:10.1016/j.bmcl.2011.06.035

Aruncus dioicus (708 words) [view diff] exact match in snippet view article find links to article

Kamtschaticus and their antioxidant and cytotoxic activities". Bioorganic & Medicinal Chemistry Letters. 21 (11): 3252–3256. doi:10.1016/j.bmcl.2011.04.043

JWH-251 (254 words) [view diff] exact match in snippet view article find links to article

"1-Pentyl-3-phenylacetylindoles, a new class of cannabimimetic indoles". Bioorganic & Medicinal Chemistry Letters. 15 (18): 4110–3. doi:10.1016/j.bmcl.2005.06.008. PMID 16005223

JWH-424 (181 words) [view diff] exact match in snippet view article find links to article

electronic effects of 4- and 8-halogenated naphthoyl substituents". Bioorganic & Medicinal Chemistry. 20 (6): 2067–81. doi:10.1016/j.bmc.2012.01.038. PMC 3298571

Vixotrigine (221 words) [view diff] exact match in snippet view article find links to article

"Recent progress in sodium channel modulators for pain". Bioorganic & Medicinal Chemistry Letters. 24 (16): 3690–3699. doi:10.1016/j.bmcl.2014.06.038

JWH-167 (183 words) [view diff] exact match in snippet view article find links to article

"1-Pentyl-3-phenylacetylindoles, a new class of cannabimimetic indoles". Bioorganic & Medicinal Chemistry Letters. 15 (18): 4110–3. doi:10.1016/j.bmcl.2005.06.008. PMID 16005223

JWH-307 (242 words) [view diff] exact match in snippet view article find links to article

affinity ligands for the cannabinoid CB1 and CB2 receptors. Bioorganic & Medicinal Chemistry Letters 2006; 16:5432-5435. Ernst L, Krüger K, Lindigkeit R

JWH-147 (203 words) [view diff] exact match in snippet view article find links to article

affinity ligands for the cannabinoid CB1 and CB2 receptors". Bioorganic & Medicinal Chemistry Letters. 16 (20): 5432–5. doi:10.1016/j.bmcl.2006.07.051. PMID 16889960

JWH-148 (169 words) [view diff] exact match in snippet view article find links to article

substituents. New highly selective CB(2) receptor agonists". Bioorganic & Medicinal Chemistry. 13 (1): 89–112. doi:10.1016/j.bmc.2004.09.050. PMID 15582455

JWH-149 (173 words) [view diff] exact match in snippet view article find links to article

substituents. New highly selective CB(2) receptor agonists". Bioorganic & Medicinal Chemistry. 13 (1): 89–112. doi:10.1016/j.bmc.2004.09.050. PMID 15582455

PHA-57378 (139 words) [view diff] exact match in snippet view article find links to article

4]diazepino[1,7-a]indoles: new templates for 5-HT(2C) agonists". Bioorganic & Medicinal Chemistry Letters. 13 (14): 2369–72. doi:10.1016/S0960-894X(03)00403-7

Topological index (1,228 words) [view diff] exact match in snippet view article find links to article

to Vibrio fischeri using genetic function approximation". Bioorganic & Medicinal Chemistry. 13 (4): 1185–94. doi:10.1016/j.bmc.2004.11.014. PMID 15670927

PNU-181731 (166 words) [view diff] exact match in snippet view article find links to article

4]diazepino[1,7-a]indoles: new templates for 5-HT(2C) agonists". Bioorganic & Medicinal Chemistry Letters. 13 (14): 2369–72. doi:10.1016/S0960-894X(03)00403-7

LY-456219 (152 words) [view diff] exact match in snippet view article find links to article

antagonist/serotonin reuptake inhibitor lead using rapid parallel synthesis". Bioorganic & Medicinal Chemistry Letters. 14 (10): 2469–2472. doi:10.1016/j.bmcl.2004.03.003

Unspecific peroxygenase (473 words) [view diff] exact match in snippet view article find links to article

5-hydroxypropranolol and 4'-hydroxydiclofenac with a fungal peroxygenase". Bioorganic & Medicinal Chemistry Letters. 19 (11): 3085–7. doi:10.1016/j.bmcl.2009.04.015. PMID 19394224

Discovery and development of ACE inhibitors (3,409 words) [view diff] exact match in snippet view article find links to article

domain-selective angiotensin I-converting enzyme inhibitors", Bioorganic & Medicinal Chemistry Letters, 16 (17): 4612–4615, doi:10.1016/j.bmcl.2006.06.003

BRL-32872 (812 words) [view diff] exact match in snippet view article find links to article

agents with potassium and calcium channel blocking properties. Bioorganic & Medicinal Chemistry, 6(11), 1993-2011 Guyton, Arthur C., Hall, John E. (2006).

Ancistrocladus korupensis (634 words) [view diff] exact match in snippet view article find links to article

the tetrahydroisoquinoline rings for biological activity". Bioorganic & Medicinal Chemistry Letters. 7 (1): 2687–2690. doi:10.1016/S0960-894X(97)10057-9

JWH-249 (193 words) [view diff] exact match in snippet view article find links to article

"1-Pentyl-3-phenylacetylindoles, a new class of cannabimimetic indoles". Bioorganic & Medicinal Chemistry Letters. 15 (18): 4110–3. doi:10.1016/j.bmcl.2005.06.008. PMID 16005223

JWH-120 (175 words) [view diff] exact match in snippet view article find links to article

substituents. New highly selective CB(2) receptor agonists". Bioorganic & Medicinal Chemistry. 13 (1): 89–112. doi:10.1016/j.bmc.2004.09.050. PMID 15582455

WAY-317538 (201 words) [view diff] exact match in snippet view article find links to article

SEN12333/WAY-317538: Novel alpha 7 nicotinic acetylcholine receptor agonist". Bioorganic & Medicinal Chemistry. 17 (14): 5247–58. doi:10.1016/j.bmc.2009.05.040. PMID 19515567

JWH-359 (165 words) [view diff] exact match in snippet view article find links to article

new selective ligands for the CB2 receptor". Bioorganic & Medicinal Chemistry. 14 (1): 247–62. doi:10.1016/j.bmc.2005.08.013. PMID 16165365

Cobalt-precorrin-7 (C15)-methyltransferase (decarboxylating) (220 words) [view diff] exact match in snippet view article

synthesized by enzymes of the vitamin B12 anaerobic pathway". Bioorganic & Medicinal Chemistry. 14 (3): 724–31. doi:10.1016/j.bmc.2005.08.062. PMID 16198574

DR-4485 (133 words) [view diff] exact match in snippet view article find links to article

antagonists with increased In vitro metabolic stability". Bioorganic & Medicinal Chemistry Letters. 13 (1): 61–4. doi:10.1016/s0960-894x(02)00842-9. PMID 12467617

JWH-302 (207 words) [view diff] exact match in snippet view article find links to article

"1-Pentyl-3-phenylacetylindoles, a new class of cannabimimetic indoles". Bioorganic & Medicinal Chemistry Letters. 15 (18): 4110–3. doi:10.1016/j.bmcl.2005.06.008. PMID 16005223

Gp41 (1,709 words) [view diff] exact match in snippet view article find links to article

"Enhanced potency of bivalent small molecule gp41 inhibitors". Bioorganic & Medicinal Chemistry. 25 (1): 408–420. doi:10.1016/j.bmc.2016.11.010. PMC 5260928

IDRA-21 (769 words) [view diff] exact match in snippet view article find links to article

subgroup of AMPA receptor modulators with improved affinity". Bioorganic & Medicinal Chemistry. 10 (5): 1229–48. CiteSeerX 10.1.1.113.7845. doi:10

Rocaglamide (373 words) [view diff] exact match in snippet view article find links to article

advances in the biology and chemistry of the flavaglines". Bioorganic & Medicinal Chemistry. 20 (6): 1857–64. doi:10.1016/j.bmc.2011.10.048. PMID 22071525

LY-456220 (152 words) [view diff] exact match in snippet view article find links to article

antagonist/serotonin reuptake inhibitor lead using rapid parallel synthesis". Bioorganic & Medicinal Chemistry Letters. 14 (10): 2469–72. doi:10.1016/j.bmcl.2004.03.003.

Α-Fluoromethylhistidine (518 words) [view diff] exact match in snippet view article find links to article

of its efficacy as a glutathione S-transferase inhibitor". Bioorganic & Medicinal Chemistry Letters. 27 (6): 1335–1340. doi:10.1016/j.bmcl.2017.02.024

David A. Evans (826 words) [view diff] exact match in snippet view article find links to article

"Tetrahedron Prize for Creativity in Organic Chemistry or Bioorganic & Medicinal Chemistry". Elsevier. Archived from the original on September 9, 2014

Jadomycin (901 words) [view diff] exact match in snippet view article find links to article

jadomycins: incorporation of non-natural and natural amino acids". Bioorganic & Medicinal Chemistry Letters. 15 (5): 1447–1449. doi:10.1016/j.bmcl.2004.12.082

Aureusidin synthase (1,400 words) [view diff] exact match in snippet view article find links to article

antioxidant and soybean lipoxygenase inhibitory activity". Bioorganic & Medicinal Chemistry. 17 (23): 8073–85. doi:10.1016/j.bmc.2009.10.002. PMID 19853459

David A. Evans (826 words) [view diff] exact match in snippet view article find links to article

"Tetrahedron Prize for Creativity in Organic Chemistry or Bioorganic & Medicinal Chemistry". Elsevier. Archived from the original on September 9, 2014

Vesicular monoamine transporter 2 (2,778 words) [view diff] exact match in snippet view article find links to article

analogs as potent inhibitors of vesicular [3H]dopamine uptake". Bioorganic & Medicinal Chemistry. 21 (21): 6771–6777. doi:10.1016/j.bmc.2013.08.001. Vartak

Α-Glucosidase (1,748 words) [view diff] exact match in snippet view article find links to article

of novel flavonoid alkaloids as α-glucosidase inhibitors". Bioorganic & Medicinal Chemistry. 25 (20): 5355–64. doi:10.1016/j.bmc.2017.07.055. PMID 28797772

Qubit fluorometer (672 words) [view diff] exact match in snippet view article find links to article

DNA-binding agents using topoisomerase I DNA unwinding assay". Bioorganic & Medicinal Chemistry Letters. 17 (4): 1013–1017. doi:10.1016/j.bmcl.2006.11.038

Dendrobium nobile (838 words) [view diff] exact match in snippet view article find links to article

production of nitric oxide in macrophage RAW 264.7 cells". Bioorganic & Medicinal Chemistry Letters. 20 (12): 3785–7. doi:10.1016/j.bmcl.2010.04.054. PMID 20483604

Tambjamine (661 words) [view diff] exact match in snippet view article find links to article

tambjamine alkaloid from the Azorean nudibranch Tambja ceutae". Bioorganic & Medicinal Chemistry Letters. 20 (8): 2668–2670. doi:10.1016/j.bmcl.2010.02.020

JWH-373 (243 words) [view diff] exact match in snippet view article find links to article

affinity ligands for the cannabinoid CB1 and CB2 receptors". Bioorganic & Medicinal Chemistry Letters. 16 (20): 5432–5. doi:10.1016/j.bmcl.2006.07.051. PMID 16889960

Arame (716 words) [view diff] exact match in snippet view article find links to article

phlorotannins from Eisenia bicyclis with BACE1 inhibitory activity". Bioorganic & Medicinal Chemistry Letters. 20 (11): 3211–5. doi:10.1016/j.bmcl.2010.04.093. PMID 20462757

Sponge isolates (883 words) [view diff] exact match in snippet view article find links to article

inhibitor isolated from a Vanuatu marine sponge Xestospongia sp". Bioorganic & Medicinal Chemistry. 14 (13): 4477–4482. doi:10.1016/j.bmc.2006.02.026. ISSN 0968-0896

JWH-145 (253 words) [view diff] exact match in snippet view article find links to article

affinity ligands for the cannabinoid CB1 and CB2 receptors". Bioorganic & Medicinal Chemistry Letters. 16 (20): 5432–5. doi:10.1016/j.bmcl.2006.07.051. PMID 16889960

Vornorexant (390 words) [view diff] exact match in snippet view article find links to article

orexin 1/2 receptor antagonist for the treatment of insomnia". Bioorganic & Medicinal Chemistry. 28 (13): 115489. doi:10.1016/j.bmc.2020.115489. PMID 32482533

JWH-369 (245 words) [view diff] exact match in snippet view article find links to article

affinity ligands for the cannabinoid CB1 and CB2 receptors". Bioorganic & Medicinal Chemistry Letters. 16 (20): 5432–5. doi:10.1016/j.bmcl.2006.07.051. PMID 16889960

Sodium channel blocker (1,207 words) [view diff] exact match in snippet view article find links to article

"Recent progress in sodium channel modulators for pain". Bioorganic & Medicinal Chemistry Letters. 24 (16): 3690–9. doi:10.1016/j.bmcl.2014.06.038. ISSN 0960-894X

S-444,823 (140 words) [view diff] exact match in snippet view article find links to article

a potent CB1/CB2 dual agonist as an antipruritic agent". Bioorganic & Medicinal Chemistry Letters. 22 (8): 2898–901. doi:10.1016/j.bmcl.2012.02.050.

JWH-309 (245 words) [view diff] exact match in snippet view article find links to article

affinity ligands for the cannabinoid CB1 and CB2 receptors". Bioorganic & Medicinal Chemistry Letters. 16 (20): 5432–5. doi:10.1016/j.bmcl.2006.07.051. PMID 16889960

XL-413 (248 words) [view diff] exact match in snippet view article find links to article

"Discovery of XL413, a potent and selective CDC7 inhibitor". Bioorganic & Medicinal Chemistry Letters. 22 (11): 3727–31. doi:10.1016/j.bmcl.2012.04.024.

JWH-363 (248 words) [view diff] exact match in snippet view article find links to article

affinity ligands for the cannabinoid CB1 and CB2 receptors". Bioorganic & Medicinal Chemistry Letters. 16 (20): 5432–5. doi:10.1016/j.bmcl.2006.07.051. PMID 16889960

PTI-1 (173 words) [view diff] exact match in snippet view article find links to article

bioavailable heterocycle-based cannabinoid CB1 receptor agonists". Bioorganic & Medicinal Chemistry Letters. 21 (6): 1748–53. doi:10.1016/j.bmcl.2011.01.082. PMID 21316962

CPP-115 (358 words) [view diff] exact match in snippet view article find links to article

novel heteroaromatic substrates of GABA aminotransferase". Bioorganic & Medicinal Chemistry. 20 (19): 5763–5773. doi:10.1016/j.bmc.2012.08.009. PMC 3448830

JWH-164 (237 words) [view diff] exact match in snippet view article find links to article

substituents. New highly selective CB(2) receptor agonists". Bioorganic & Medicinal Chemistry. 13 (1): 89–112. doi:10.1016/j.bmc.2004.09.050. PMID 15582455

CYP1B1 (1,185 words) [view diff] exact match in snippet view article find links to article

"A new class of CYP1B1 inhibitors derived from bentranil". Bioorganic & Medicinal Chemistry Letters. 80: 129112. doi:10.1016/j.bmcl.2022.129112. Smith

MCHB-1 (218 words) [view diff] exact match in snippet view article find links to article

"Novel benzimidazole derivatives as selective CB2 agonists". Bioorganic & Medicinal Chemistry Letters. 18 (13): 3695–700. doi:10.1016/j.bmcl.2008.05.073

Raymond Lemieux (861 words) [view diff] exact match in snippet view article find links to article

Hindsgaul, O.; Bundle, D. R. (1996). "Raymond U. Lemieux". Bioorganic & Medicinal Chemistry. 4 (11): 1795–1797. doi:10.1016/S0968-0896(96)00245-3. PMID 9007264

RQ-00202730 (193 words) [view diff] exact match in snippet view article find links to article

RQ-00202730, for the treatment of irritable bowel syndrome". Bioorganic & Medicinal Chemistry Letters. 25 (2): 236–40. doi:10.1016/j.bmcl.2014.11.062. PMID 25499880

BMS-F (197 words) [view diff] exact match in snippet view article find links to article

2002). "C-3 Amido-indole cannabinoid receptor modulators". Bioorganic & Medicinal Chemistry Letters. 12 (17): 2399–2402. doi:10.1016/s0960-894x(02)00466-3

JWH-366 (251 words) [view diff] exact match in snippet view article find links to article

affinity ligands for the cannabinoid CB1 and CB2 receptors". Bioorganic & Medicinal Chemistry Letters. 16 (20): 5432–5. doi:10.1016/j.bmcl.2006.07.051. PMID 16889960

Dawn Ward (chemist) (225 words) [view diff] exact match in snippet view article

analogs are potent inhibitors of hepatitis C virus replication". Bioorganic & Medicinal Chemistry Letters. 24 (2): 609–612. doi:10.1016/j.bmcl.2013.12.012. ISSN 0960-894X

PNU-282,987 (396 words) [view diff] exact match in snippet view article find links to article

amides as alpha7 nicotinic acetylcholine receptor agonists". Bioorganic & Medicinal Chemistry. 14 (24): 8219–8248. doi:10.1016/j.bmc.2006.09.019. PMID 17011782

JWH-368 (252 words) [view diff] exact match in snippet view article find links to article

affinity ligands for the cannabinoid CB1 and CB2 receptors". Bioorganic & Medicinal Chemistry Letters. 16 (20): 5432–5. doi:10.1016/j.bmcl.2006.07.051. PMID 16889960

JWH-367 (250 words) [view diff] exact match in snippet view article find links to article

affinity ligands for the cannabinoid CB1 and CB2 receptors". Bioorganic & Medicinal Chemistry Letters. 16 (20): 5432–5. doi:10.1016/j.bmcl.2006.07.051. PMID 16889960

Alniditan (341 words) [view diff] exact match in snippet view article find links to article

"The discovery of a series of new non-indole 5HT1D agonists". Bioorganic & Medicinal Chemistry Letters. 5 (22): 2649–2654. doi:10.1016/0960-894X(95)00473-7

FUBIMINA (347 words) [view diff] exact match in snippet view article find links to article

"Novel benzimidazole derivatives as selective CB2 agonists". Bioorganic & Medicinal Chemistry Letters. 18 (13): 3695–3700. doi:10.1016/j.bmcl.2008.05.073

JWH-098 (355 words) [view diff] exact match in snippet view article find links to article

substituents. New highly selective CB(2) receptor agonists". Bioorganic & Medicinal Chemistry. 13 (1): 89–112. doi:10.1016/j.bmc.2004.09.050. PMID 15582455

EPPTB (652 words) [view diff] exact match in snippet view article find links to article

amine-associated receptor 1 (mTAAR1): discovery of EPPTB (RO5212773)". Bioorganic & Medicinal Chemistry Letters. 21 (4): 1227–31. doi:10.1016/j.bmcl.2010.12.075. PMID 21237643

Estrone phosphate (211 words) [view diff] exact match in snippet view article find links to article

sulfatase with 4-substituted estrone and estradiol derivatives". Bioorganic & Medicinal Chemistry. 19 (20): 5999–6005. doi:10.1016/j.bmc.2011.08.046. PMID 21925885

Pesticide research (1,397 words) [view diff] exact match in snippet view article find links to article

(June 2009). "Combinatorial chemistry in the agrosciences". Bioorganic & Medicinal Chemistry. 17 (12): 4035–46. doi:10.1016/j.bmc.2009.03.027. PMID 19349185

JWH-365 (254 words) [view diff] exact match in snippet view article find links to article

affinity ligands for the cannabinoid CB1 and CB2 receptors". Bioorganic & Medicinal Chemistry Letters. 16 (20): 5432–5. doi:10.1016/j.bmcl.2006.07.051. PMID 16889960

JWH-370 (252 words) [view diff] exact match in snippet view article find links to article

affinity ligands for the cannabinoid CB1 and CB2 receptors". Bioorganic & Medicinal Chemistry Letters. 16 (20): 5432–5. doi:10.1016/j.bmcl.2006.07.051. PMID 16889960

JWH-146 (255 words) [view diff] exact match in snippet view article find links to article

affinity ligands for the cannabinoid CB1 and CB2 receptors". Bioorganic & Medicinal Chemistry Letters. 16 (20): 5432–5. doi:10.1016/j.bmcl.2006.07.051. PMID 16889960

Bicyclomycin (839 words) [view diff] exact match in snippet view article find links to article

dihydrobicyclomycins: synthesis and biochemical and biological properties". Bioorganic & Medicinal Chemistry. 14 (1): 41–61. doi:10.1016/j.bmc.2005.07.075. PMID 16185879

Viminol (641 words) [view diff] exact match in snippet view article find links to article

stereoisomers of Z4349, a novel and selective μ-opioid analgesic". Bioorganic & Medicinal Chemistry Letters. 6 (5): 589–592. doi:10.1016/0960-894X(95)00077-7.

JWH-364 (245 words) [view diff] exact match in snippet view article find links to article

affinity ligands for the cannabinoid CB1 and CB2 receptors". Bioorganic & Medicinal Chemistry Letters. 16 (20): 5432–5. doi:10.1016/j.bmcl.2006.07.051. PMID 16889960

Piclozotan (170 words) [view diff] exact match in snippet view article find links to article

agonists with neuroprotective effect: Discovery of Piclozotan". Bioorganic & Medicinal Chemistry. 14 (6): 1978–92. doi:10.1016/j.bmc.2005.10.046. PMID 16290165

Mixed inhibition (1,086 words) [view diff] exact match in snippet view article find links to article

fukugetin as a mixed-type inhibitor for human tissue kallikreins". Bioorganic & Medicinal Chemistry Letters. 26 (5): 1485–1489. doi:10.1016/j.bmcl.2016.01.039

Pacific Blue (dye) (370 words) [view diff] exact match in snippet view article

Coumarins: Excellent UV-Light Excitable Fluorescent Dyes". Bioorganic & Medicinal Chemistry Letters. 8 (1): 3107–3110. doi:10.1016/s0960-894x(98)00578-2

2-Benzylpiperidine (749 words) [view diff] exact match in snippet view article find links to article

"Probing the proposed phenyl-A region of the sigma-1 receptor". Bioorganic & Medicinal Chemistry. 10 (8): 2759–2765. doi:10.1016/S0968-0896(02)00096-2. PMID 12057665

S-777,469 (243 words) [view diff] exact match in snippet view article find links to article

an orally available CB2 agonist as an antipruritic agent". Bioorganic & Medicinal Chemistry Letters. 22 (8): 2803–6. doi:10.1016/j.bmcl.2012.02.072. PMID 22444677

GPR119 (1,172 words) [view diff] exact match in snippet view article find links to article

"2,5-Disubstituted pyridines as potent GPR119 agonists". Bioorganic & Medicinal Chemistry Letters. 20 (8): 2577–2581. doi:10.1016/j.bmcl.2010.02.083

LY-341495 (1,011 words) [view diff] exact match in snippet view article find links to article

acid and its 6-heptyl ester, a potent mGluR2 antagonist". Bioorganic & Medicinal Chemistry. 16 (8): 4359–66. doi:10.1016/j.bmc.2008.02.066. PMID 18348906

In'oya (629 words) [view diff] exact match in snippet view article find links to article

spider venom: A novel class of melanogenesis inhibitors". Bioorganic & Medicinal Chemistry. 24 (22): 5685–5692. doi:10.1016/j.bmc.2016.08.023. PMID 27647371

Minimal infective dose (1,288 words) [view diff] exact match in snippet view article find links to article

characterize antimicrobial compounds through kinetic dose response". Bioorganic & Medicinal Chemistry. 24 (24): 6315–6319. doi:10.1016/j.bmc.2016.09.053. ISSN 1464-3391

Ro60-0213 (263 words) [view diff] exact match in snippet view article find links to article

3-g]indazol-1-yl)ethylamine derivatives as 5-HT2C receptor agonists". Bioorganic & Medicinal Chemistry. 16 (4): 1966–82. doi:10.1016/j.bmc.2007.10.100. PMID 18035544

2-Imidazoline (902 words) [view diff] exact match in snippet view article find links to article

inhibitors: Design, synthesis, and biological evaluation". Bioorganic & Medicinal Chemistry Letters. 29 (16): 2364–2368. doi:10.1016/j.bmcl.2019.06.007

5-Benzyloxytryptamine (255 words) [view diff] exact match in snippet view article find links to article

2010). "5-benzyloxytryptamine as an antagonist of TRPM8". Bioorganic & Medicinal Chemistry Letters. 20 (23): 7076–7079. doi:10.1016/j.bmcl.2010.09.099

Cortinarius infractus (932 words) [view diff] exact match in snippet view article find links to article

"Acetylcholinesterase inhibitors from the toadstool Cortinarius infractus". Bioorganic & Medicinal Chemistry. 18 (6): 2173–77. doi:10.1016/j.bmc.2010.01.074. PMID 20176490

Tropinone (1,032 words) [view diff] exact match in snippet view article find links to article

ketones as a novel class of dopamine transporter inhibitors". Bioorganic & Medicinal Chemistry. 9 (7): 1753–1764. doi:10.1016/S0968-0896(01)00090-6. PMID 11425577

2-Benzylpiperidine (749 words) [view diff] exact match in snippet view article find links to article

"Probing the proposed phenyl-A region of the sigma-1 receptor". Bioorganic & Medicinal Chemistry. 10 (8): 2759–2765. doi:10.1016/S0968-0896(02)00096-2. PMID 12057665

List of methylphenidate analogues (2,336 words) [view diff] exact match in snippet view article find links to article

evaluation, and dopamine transporter photoaffinity labeling". Bioorganic & Medicinal Chemistry. 19 (1): 504–12. doi:10.1016/j.bmc.2010.11.002. PMC 3023924

JWH-122 (375 words) [view diff] exact match in snippet view article find links to article

substituents. New highly selective CB(2) receptor agonists". Bioorganic & Medicinal Chemistry. 13 (1): 89–112. doi:10.1016/j.bmc.2004.09.050. PMID 15582455

Magnolol (661 words) [view diff] exact match in snippet view article find links to article

honokiol as potent allosteric potentiators of GABAA receptors". Bioorganic & Medicinal Chemistry. 22 (24): 6908–6917. doi:10.1016/j.bmc.2014.10.027. PMID 25456080

Brain positron emission tomography (1,867 words) [view diff] exact match in snippet view article find links to article

positron emission tomography (PET) imaging of amyloid in brain". Bioorganic & Medicinal Chemistry Letters. 12 (3): 295–8. doi:10.1016/S0960-894X(01)00734-X.

Shankar Balasubramanian (1,401 words) [view diff] exact match in snippet view article find links to article

<"Tetrahedron Prize for Creativity in Organic Chemistry or Bioorganic & Medicinal Chemistry | Elsevier". Archived from the original on 9 September 2014

Retosiban (1,099 words) [view diff] exact match in snippet view article find links to article

of GSK221149A: a potent and selective oxytocin antagonist". Bioorganic & Medicinal Chemistry Letters. 18 (1): 90–4. doi:10.1016/j.bmcl.2007.11.008. PMID 18032036

3CLpro-1 (426 words) [view diff] exact match in snippet view article find links to article

of 3C protease inhibitors as anti-enterovirus 71 agents". Bioorganic & Medicinal Chemistry. 16 (15): 7388–98. doi:10.1016/j.bmc.2008.06.015. PMC 7125518

TRPA (ion channel) (809 words) [view diff] exact match in snippet view article

non-electrophilic reference agonist of the TrpA1 channel". Bioorganic & Medicinal Chemistry Letters. 21 (16): 4857–9. doi:10.1016/j.bmcl.2011.06.035. PMID 21741838

Regorafenib (936 words) [view diff] exact match in snippet view article find links to article

evaluation of sorafenib- and regorafenib-like sEH inhibitors". Bioorganic & Medicinal Chemistry Letters. 23 (13): 3732–7. doi:10.1016/j.bmcl.2013.05.011. PMC 3744640

Fatty acid synthase (4,020 words) [view diff] exact match in snippet view article find links to article

acylphloroglucinols isolated from Dryopteris crassirhizoma". Bioorganic & Medicinal Chemistry Letters. 16 (18): 4738–4742. doi:10.1016/j.bmcl.2006.07.018

Duranta erecta (1,257 words) [view diff] exact match in snippet view article find links to article

antioxidative coumarinolignoids from Duranta repens Linn". Bioorganic & Medicinal Chemistry Letters. 19 (13): 3521–3524. doi:10.1016/j.bmcl.2009.05.006

Differentiation-inducing factor (1,062 words) [view diff] exact match in snippet view article find links to article

derivatives that selectively suppress innate immune responses". Bioorganic & Medicinal Chemistry. 23 (15): 4311–4315. doi:10.1016/j.bmc.2015.06.027. PMID 26122773

Gould–Jacobs reaction (752 words) [view diff] exact match in snippet view article find links to article

pyrazoloquinolin-3-ones: synthesis and in vitro BZR activity". Bioorganic & Medicinal Chemistry. 13 (10): 3531–3541. doi:10.1016/j.bmc.2005.02.042. PMID 15848766

AMG-3 (353 words) [view diff] exact match in snippet view article find links to article

novel cannabinoid ligands with optimum binding activity". Bioorganic & Medicinal Chemistry Letters. 17 (24): 6754–63. doi:10.1016/j.bmcl.2007.10.044.

Nutlin (603 words) [view diff] exact match in snippet view article find links to article

inhibitors: Design, synthesis, and biological evaluation". Bioorganic & Medicinal Chemistry Letters. 29 (16): 2364–2368. doi:10.1016/j.bmcl.2019.06.007

JWH-371 (253 words) [view diff] exact match in snippet view article find links to article

affinity ligands for the cannabinoid CB1 and CB2 receptors". Bioorganic & Medicinal Chemistry Letters. 16 (20): 5432–5. doi:10.1016/j.bmcl.2006.07.051. PMID 16889960

Sufugolix (562 words) [view diff] exact match in snippet view article find links to article

3-d]pyrimidine-2,4-diones as human GnRH receptor antagonists". Bioorganic & Medicinal Chemistry. 15 (16): 5590–5603. doi:10.1016/j.bmc.2007.05.029. PMID 17561404

JWH-372 (289 words) [view diff] exact match in snippet view article find links to article

affinity ligands for the cannabinoid CB1 and CB2 receptors". Bioorganic & Medicinal Chemistry Letters. 16 (20): 5432–5. doi:10.1016/j.bmcl.2006.07.051. PMID 16889960

JWH-150 (249 words) [view diff] exact match in snippet view article find links to article

affinity ligands for the cannabinoid CB1 and CB2 receptors". Bioorganic & Medicinal Chemistry Letters. 16 (20): 5432–5. doi:10.1016/j.bmcl.2006.07.051. PMID 16889960

3-Phenylcoumarin (294 words) [view diff] exact match in snippet view article find links to article

"New halogenated phenylcoumarins as tyrosinase inhibitors". Bioorganic & Medicinal Chemistry Letters. 21 (11): 3342–3345. doi:10.1016/j.bmcl.2011.04.012

Alan R. Katritzky (1,200 words) [view diff] exact match in snippet view article find links to article

2006). "QSAR study of mosquito repellents using Codessa Pro". Bioorganic & Medicinal Chemistry Letters. 16 (8): 2306–2311. doi:10.1016/j.bmcl.2005.11.113

Mesotrione (1,595 words) [view diff] exact match in snippet view article find links to article

the triketone chemistry story from a Syngenta perspective". Bioorganic & Medicinal Chemistry. 17 (12): 4134–4152. doi:10.1016/j.bmc.2009.03.015. PMID 19349184

PTI-2 (175 words) [view diff] exact match in snippet view article find links to article

bioavailable heterocycle-based cannabinoid CB1 receptor agonists". Bioorganic & Medicinal Chemistry Letters. 21 (6): 1748–53. doi:10.1016/j.bmcl.2011.01.082. PMID 21316962

JWH-203 (458 words) [view diff] exact match in snippet view article find links to article

"1-Pentyl-3-phenylacetylindoles, a new class of cannabimimetic indoles". Bioorganic & Medicinal Chemistry Letters. 15 (18): 4110–3. doi:10.1016/j.bmcl.2005.06.008. PMID 16005223

1,2-Dioxolane (720 words) [view diff] exact match in snippet view article find links to article

2-dioxolanes and their activity against Plasmodium falciparum". Bioorganic & Medicinal Chemistry Letters. 18 (24): 6521–4. doi:10.1016/j.bmcl.2008.10.083. PMID 18993067

RCS-8 (197 words) [view diff] exact match in snippet view article find links to article

"Design, Synthesis and Pharmacology of Cannabimimetic Indoles". Bioorganic & Medicinal Chemistry Letters. 4 (4): 563–566. doi:10.1016/S0960-894X(01)80155-4

DAA-1106 (611 words) [view diff] exact match in snippet view article find links to article

derivatives as novel peripheral benzodiazepine receptor ligands". Bioorganic & Medicinal Chemistry. 12 (2): 423–38. doi:10.1016/j.bmc.2003.10.050. PMID 14723961

BIM-018 (115 words) [view diff] exact match in snippet view article find links to article

"Novel benzimidazole derivatives as selective CB2 agonists". Bioorganic & Medicinal Chemistry Letters. 18 (13): 3695–700. doi:10.1016/j.bmcl.2008.05.073

Lactase (2,113 words) [view diff] exact match in snippet view article find links to article

their use in the evaluation of lactase activity in vivo". Bioorganic & Medicinal Chemistry. 15 (14): 4836–40. doi:10.1016/j.bmc.2007.04.067. hdl:10261/81580

LR-5182 (455 words) [view diff] exact match in snippet view article find links to article

triple re-uptake inhibitors for the treatment of depression". Bioorganic & Medicinal Chemistry Letters. 13 (19): 3277–80. doi:10.1016/S0960-894X(03)00660-7

2F-QMPSB (291 words) [view diff] exact match in snippet view article find links to article

CB2 receptor agonists for the treatment of chronic pain". Bioorganic & Medicinal Chemistry Letters. 21 (1): 182–5. doi:10.1016/j.bmcl.2010.11.044. PMID 21115245

O-1269 (380 words) [view diff] exact match in snippet view article find links to article

unique binding selectivities and pharmacological activities". Bioorganic & Medicinal Chemistry. 13 (18): 5463–74. doi:10.1016/j.bmc.2005.06.005. PMID 15994087

Cytokinin (1,978 words) [view diff] exact match in snippet view article find links to article

Spíchal L (February 2016). "Use of cytokinins as agrochemicals". Bioorganic & Medicinal Chemistry. Recent Developments in Agrochemistry. 24 (3): 484–492. doi:10

Substituted tryptamine (2,080 words) [view diff] exact match in snippet view article find links to article

"Alpha-ethyltryptamines as dual dopamine-serotonin releasers". Bioorganic & Medicinal Chemistry Letters. 24 (19): 4754–4758. doi:10.1016/j.bmcl.2014.07.062

CSP-2503 (229 words) [view diff] exact match in snippet view article find links to article

using computational simulation. A 5-HT1A receptor agonist". Bioorganic & Medicinal Chemistry Letters. 13 (8): 1429–32. doi:10.1016/S0960-894X(03)00160-4

AM-630 (472 words) [view diff] exact match in snippet view article find links to article

2002). "C-3 Amido-indole cannabinoid receptor modulators". Bioorganic & Medicinal Chemistry Letters. 12 (17): 2399–2402. doi:10.1016/S0960-894X(02)00466-3

AM-1220 (485 words) [view diff] exact match in snippet view article find links to article

"C-Attached aminoalkylindoles: potent cannabinoid mimetics". Bioorganic & Medicinal Chemistry Letters. 6 (1): 17–22. doi:10.1016/0960-894X(95)00560-G. Deng

Alendronic acid (1,175 words) [view diff] exact match in snippet view article find links to article

drugs--reports of new drugs recently approved by the FDA. Alendronate". Bioorganic & Medicinal Chemistry. 4 (1): 3–4. doi:10.1016/0968-0896(96)00042-9. PMID 8689235

Seviteronel (882 words) [view diff] exact match in snippet view article find links to article

4-(1,2,3-triazole)-based P450c17a 17,20-lyase inhibitors". Bioorganic & Medicinal Chemistry Letters. 24 (11): 2444–2447. doi:10.1016/j.bmcl.2014.04.024

List of 5α-reductase inhibitors (3,041 words) [view diff] exact match in snippet view article find links to article

"Ganoderic acid DM: anti-androgenic osteoclastogenesis inhibitor". Bioorganic & Medicinal Chemistry Letters. 19 (8): 2154–7. doi:10.1016/j.bmcl.2009.02.119. PMID 19289282

Pandanus utilis (1,286 words) [view diff] case mismatch in snippet view article find links to article

(2005). Biology of Plants, 7th ed. W.H. Freeman and Company. "Bioorganic & medicinal chemistry letters". D.L. Tomlinson "A Leaf and Fruit Disease of Pandanus

Alendronic acid (1,175 words) [view diff] exact match in snippet view article find links to article

drugs--reports of new drugs recently approved by the FDA. Alendronate". Bioorganic & Medicinal Chemistry. 4 (1): 3–4. doi:10.1016/0968-0896(96)00042-9. PMID 8689235

BU72 (628 words) [view diff] exact match in snippet view article find links to article

constrained phenyl group: High affinity opioid agonists". Bioorganic & Medicinal Chemistry Letters. 5 (24): 2969–2974. doi:10.1016/0960-894X(95)00522-1

FK1012 (333 words) [view diff] exact match in snippet view article find links to article

FKBP12 ligands for the regulated dimerization of proteins". Bioorganic & Medicinal Chemistry. 6 (8): 1309–1335. doi:10.1016/S0968-0896(98)00125-4. ISSN 0968-0896

Tubulin alpha-1A chain (1,670 words) [view diff] exact match in snippet view article find links to article

may be endogenous ligands for the paclitaxel-binding site". Bioorganic & Medicinal Chemistry. 9 (8): 1967–1976. doi:10.1016/S0968-0896(01)00103-1. PMID 11504633

Furegrelate (1,892 words) [view diff] exact match in snippet view article find links to article

4-quinolones at the benzodiazepine site of GABA(A) receptors". Bioorganic & Medicinal Chemistry. 16 (14): 6936–48. doi:10.1016/j.bmc.2008.05.049. PMID 18541432

List of phenyltropanes (5,647 words) [view diff] exact match in snippet view article find links to article

discovery of a selective SERT antagonist with picomolar potency". Bioorganic & Medicinal Chemistry. 15 (4): 1131–1133. doi:10.1016/j.bmcl.2004.12.014. PMID 15686927

KvLQT1 (1,503 words) [view diff] exact match in snippet view article find links to article

and selective K(v)7.1 (KCNQ1) potassium channel activator". Bioorganic & Medicinal Chemistry Letters. 22 (18): 5936–5941. doi:10.1016/j.bmcl.2012.07.060

Peripherally acting μ-opioid receptor antagonist (3,255 words) [view diff] exact match in snippet view article find links to article

Synthesis and Computer Simulation Study". Bioorganic & Medicinal Chemistry. 25 (8): 2406–2422. doi:10.1016/j.bmc.2017.02.064. ISSN 0968-0896

Solithromycin (1,416 words) [view diff] exact match in snippet view article find links to article

2016). "The solithromycin journey-It is all in the chemistry". Bioorganic & Medicinal Chemistry. 24 (24): 6420–6428. doi:10.1016/j.bmc.2016.08.035. PMID 27595539

3-Monoacetylmorphine (191 words) [view diff] exact match in snippet view article find links to article

dihydromorphine-, and codeine 6-O-sulfate ester congeners". Bioorganic & Medicinal Chemistry Letters. 16 (16): 4291–4295. doi:10.1016/j.bmcl.2006.05.060

2-Phenylbenzofuran (417 words) [view diff] exact match in snippet view article find links to article

inhibitors: Synthesis, biological activity and molecular modeling". Bioorganic & Medicinal Chemistry Letters. 26 (9): 2308–2313. doi:10.1016/j.bmcl.2016.03.039

HBTU (639 words) [view diff] exact match in snippet view article find links to article

(1992). "HBTU: a mild activating agent of muramic acid". Bioorganic & Medicinal Chemistry Letters. 2 (6): 571–574. doi:10.1016/S0960-894X(01)81199-9

Ψ-DOM (251 words) [view diff] exact match in snippet view article find links to article

the 6-position: effects on 5-HT(2A/2C) receptor affinity". Bioorganic & Medicinal Chemistry Letters. 12 (15): 1997–9. doi:10.1016/S0960-894X(02)00306-2

Edaravone (1,629 words) [view diff] exact match in snippet view article find links to article

1-phenyl-3-methyl-5-pyrazolone (PMP), also known as edaravone". Bioorganic & Medicinal Chemistry. 28 (10): 115463. doi:10.1016/j.bmc.2020.115463. PMID 32241621

R6890 (409 words) [view diff] exact match in snippet view article find links to article

N-substituted spiropiperidines as nociceptin receptor ligands". Bioorganic & Medicinal Chemistry Letters. 17 (8): 2281–2284. doi:10.1016/j.bmcl.2007.01.069

Streptomyces nitrosporeus (722 words) [view diff] exact match in snippet view article find links to article

analogues from the marine-derived Streptomyces nitrosporeus". Bioorganic & Medicinal Chemistry Letters. 24 (22): 5288–93. doi:10.1016/j.bmcl.2014.09.049.

Racemic crystallography (1,484 words) [view diff] exact match in snippet view article find links to article

2017). "Recent advances in racemic protein crystallography". Bioorganic & Medicinal Chemistry. Peptide and protein ligation. 25 (18): 4953–4965. doi:10.1016/j

Nantenine (263 words) [view diff] exact match in snippet view article find links to article

antagonists at human 5-HT(2A) receptors: C1 and flexible congeners". Bioorganic & Medicinal Chemistry Letters. 19 (9): 2530–2. doi:10.1016/j.bmcl.2009.03.048. PMC 2677726

Alalevonadifloxacin (147 words) [view diff] exact match in snippet view article find links to article

alalevonadifloxacin for the treatment of MRSA infection". Bioorganic & Medicinal Chemistry Letters. 54: 128432. doi:10.1016/j.bmcl.2021.128432. PMID 34757217

SB-357134 (250 words) [view diff] exact match in snippet view article find links to article

4-methoxy-3-piperazin-1-ylbenzenesulfonamide (SB-357134)". Bioorganic & Medicinal Chemistry Letters. 11 (1): 55–8. doi:10.1016/S0960-894X(00)00597-7. PMID 11140733

RAR-related orphan receptor (1,127 words) [view diff] exact match in snippet view article find links to article

(2016). "Recent progress on nuclear receptor RORγ modulators". Bioorganic & Medicinal Chemistry Letters. 26 (18): 4387–93. doi:10.1016/j.bmcl.2016.08.012.

Cobicistat (913 words) [view diff] exact match in snippet view article find links to article

Part II: P2/P3 region and discovery of cobicistat (GS-9350)". Bioorganic & Medicinal Chemistry Letters. 24 (3): 995–9. doi:10.1016/j.bmcl.2013.12.057. PMID 24412072

Corepressor (2,462 words) [view diff] exact match in snippet view article find links to article

interaction inhibitor by utilizing structure-based drug design". Bioorganic & Medicinal Chemistry. 25 (17): 4876–4886. doi:10.1016/j.bmc.2017.07.037. PMID 28760529

Neuraminidase (1,568 words) [view diff] exact match in snippet view article find links to article

Part 1: selective inhibitors of lysosomal sialidase (NEU1)". Bioorganic & Medicinal Chemistry Letters. 18 (2): 532–7. doi:10.1016/j.bmcl.2007.11.084. PMID 18068975

JWH-210 (500 words) [view diff] exact match in snippet view article find links to article

substituents. New highly selective CB(2) receptor agonists". Bioorganic & Medicinal Chemistry. 13 (1): 89–112. doi:10.1016/j.bmc.2004.09.050. PMID 15582455

Copalic acid (349 words) [view diff] exact match in snippet view article find links to article

down-regulate androgen receptor and inhibit small chaperone protein". Bioorganic & Medicinal Chemistry Letters. 27 (11): 2292–2295. doi:10.1016/j.bmcl.2017.04.046

MTEP (1,514 words) [view diff] exact match in snippet view article find links to article

novel metabotropic glutamate receptor subtype 5 antagonists". Bioorganic & Medicinal Chemistry Letters. 17 (11): 2987–2991. doi:10.1016/j.bmcl.2007.03.066

EMD-386088 (218 words) [view diff] exact match in snippet view article find links to article

6-tetrahydropyridin-4-yl)-1H-indoles as novel 5-HT6 receptor agonists". Bioorganic & Medicinal Chemistry Letters. 15 (19): 4230–4234. doi:10.1016/j.bmcl.2005.06.067

SB-334867 (996 words) [view diff] exact match in snippet view article find links to article

possible confounding effects on in vivo and in vitro studies". Bioorganic & Medicinal Chemistry Letters. 22 (21): 6661–4. doi:10.1016/j.bmcl.2012.08.109. PMID 23031594

Antifungal (2,630 words) [view diff] exact match in snippet view article find links to article

(February 2017). "Antifungal activity of substituted aurones". Bioorganic & Medicinal Chemistry Letters. 27 (4): 901–903. doi:10.1016/j.bmcl.2017.01.012. PMID 28094180

Leishmania braziliensis (1,843 words) [view diff] exact match in snippet view article find links to article

Leishmania braziliensis viability and host–parasite interaction". Bioorganic & Medicinal Chemistry. 22 (21): 6220–6226. doi:10.1016/j.bmc.2014.08.023. PMID 25240731

Alpha-2B adrenergic receptor (1,754 words) [view diff] exact match in snippet view article find links to article

isolated from the Australian marine sponge, Acanthella costata". Bioorganic & Medicinal Chemistry. 17 (6): 2497–500. doi:10.1016/j.bmc.2009.01.065. hdl:10072/28568

GABAA-rho receptor (1,673 words) [view diff] exact match in snippet view article find links to article

acid at recombinant GABA(C) receptors". Bioorganic & Medicinal Chemistry Letters. 18 (1): 402–404. doi:10.1016/j.bmcl.2007.10.019. PMID 17981464

Dexoxadrol (135 words) [view diff] exact match in snippet view article find links to article

receptor antagonists derived from dexoxadrol and etoxadrol". Bioorganic & Medicinal Chemistry. 13 (24): 6836–49. doi:10.1016/j.bmc.2005.07.030. PMID 16169732

Nandina (1,551 words) [view diff] exact match in snippet view article find links to article

antagonists at human 5-HT(2A) receptors: C1 and flexible congeners". Bioorganic & Medicinal Chemistry Letters. 19 (9): 2530–2. doi:10.1016/j.bmcl.2009.03.048. PMC 2677726

RTI-126 (372 words) [view diff] exact match in snippet view article find links to article

affinities of 2- and 3-isoxazolyl-8-azabicyclo[3.2.1]octanes". Bioorganic & Medicinal Chemistry Letters. 14 (7): 1775–8. doi:10.1016/j.bmcl.2004.01.025. PMID 15026069

Dopamine releasing agent (2,007 words) [view diff] exact match in snippet view article find links to article

"Alpha-ethyltryptamines as dual dopamine-serotonin releasers". Bioorganic & Medicinal Chemistry Letters. 24 (19): 4754–4758. doi:10.1016/j.bmcl.2014.07.062

Taranabant (403 words) [view diff] exact match in snippet view article find links to article

sulfonamides as human cannabinoid-1 receptor inverse agonists". Bioorganic & Medicinal Chemistry Letters. 17 (8): 2184–7. doi:10.1016/j.bmcl.2007.01.087. PMID 17293109

Diphosphomevalonate decarboxylase (1,611 words) [view diff] exact match in snippet view article find links to article

inhibition studies of mevalonate 5-diphosphate decarboxylase". Bioorganic & Medicinal Chemistry Letters. 17 (22): 6164–6168. doi:10.1016/j.bmcl.2007.09.033

Death receptor 5 (1,534 words) [view diff] exact match in snippet view article find links to article

(IPH) that detects cancer cells and induces their apoptosis". Bioorganic & Medicinal Chemistry. 26 (17): 4804–4816. doi:10.1016/j.bmc.2018.08.016. PMID 30177492

Glycorandomization (1,507 words) [view diff] exact match in snippet view article find links to article

Thorson, J. S. (2004). "Natural product glycorandomization". Bioorganic & Medicinal Chemistry. 12 (7): 1577–1584. doi:10.1016/j.bmc.2003.12.046. PMID 15112655

Azeliragon (458 words) [view diff] exact match in snippet view article find links to article

and anti-TNBC activity of Azeliragon triazole analogues". Bioorganic & Medicinal Chemistry Letters. 54: 128444. doi:10.1016/j.bmcl.2021.128444. PMID 34763082

Zuranolone (1,167 words) [view diff] exact match in snippet view article find links to article

(2018). "Breakthroughs in neuroactive steroid drug discovery". Bioorganic & Medicinal Chemistry Letters. 28 (2): 61–70. doi:10.1016/j.bmcl.2017.11.043. PMID 29223589

Miricorilant (459 words) [view diff] exact match in snippet view article find links to article

efficacy in the olanzapine-induced weight gain model in the rat". Bioorganic & Medicinal Chemistry Letters. 22 (24): 7376–7380. doi:10.1016/j.bmcl.2012.10.074

BI 99179 (608 words) [view diff] exact match in snippet view article find links to article

inhibitor of type I fatty acid synthase with central exposure". Bioorganic & Medicinal Chemistry Letters. doi:10.1016/j.bmcl.2011.07.083. GmbH, Boehringer Ingelheim

TAS2R14 (1,957 words) [view diff] exact match in snippet view article find links to article

and selectivity of bitter molecules and their receptors". Bioorganic & Medicinal Chemistry. 23 (14): 4082–4091. doi:10.1016/j.bmc.2015.04.025. PMID 25934224

Podophyllotoxin hybrid molecule (668 words) [view diff] exact match in snippet view article find links to article

cycle arrest, binding CT DNA and inhibition of Topo IIβ". Bioorganic & Medicinal Chemistry Letters. 29 (16): 2129–2135. doi:10.1016/j.bmcl.2019.06.063

Amaryllis belladonna (815 words) [view diff] exact match in snippet view article find links to article

"Antiplasmodial alkaloids from bulbs of Amaryllis belladonna Steud". Bioorganic & Medicinal Chemistry Letters. 28 (1): 40–42. doi:10.1016/j.bmcl.2017.11.021. PMC 5753767

L-Aspartic-4-semialdehyde (624 words) [view diff] exact match in snippet view article find links to article

selective aspartate semialdehyde dehydrogenase inhibitors". Bioorganic & Medicinal Chemistry. 23 (20): 6622–6631. doi:10.1016/j.bmc.2015.09.017. PMC 4601562